Evaluation of the anticoagulant properties of aprotinin in vitro

Eur J Anaesthesiol. 1996 Sep;13(5):468-70. doi: 10.1046/j.1365-2346.1996.00991.x.

Abstract

The interaction of aprotinin with normal coagulation was studied in blood samples obtained from 10 healthy subjects. Each sample was simultaneously tested in four different preparations: NaCl-treated blood: 0.03 mL 0.9% NaCl in 0.33 mL blood; aprotinin treated blood: 0.33 mL blood+aprotinin in 0.03 mL in aliquots to obtain a final blood concentration of respectively 50 KIU mL-1; 100 KIU mL-1 and 200 KIU mL-1. The coagulation process was analysed by thromboelastography. R-time, reflecting intrinsic coagulation, increased in a dose dependent manner between NaCl-treated and aprotinin-treated blood. These findings suggest a dose dependent impairment of intrinsic coagulation by aprotinin.

MeSH terms

  • Anticoagulants / pharmacology*
  • Aprotinin / pharmacology*
  • Blood Coagulation / drug effects*
  • Dose-Response Relationship, Drug
  • Hemostatics / pharmacology*
  • Humans
  • In Vitro Techniques
  • Thrombelastography

Substances

  • Anticoagulants
  • Hemostatics
  • Aprotinin