Comparison of in vitro activities of DU-6859a and other fluoroquinolones against Japanese isolates of anaerobic bacteria

Clin Infect Dis. 1996 Dec:23 Suppl 1:S31-5. doi: 10.1093/clinids/23.supplement_1.s31.

Abstract

The in vitro activity of DU-6859a, a new fluoroquinolone, was compared with those of other fluoroquinolones against clinical isolates of anaerobic bacteria and Gardnerella vaginalis. DU-6859a was the most active agent; it inhibited 90% of isolates of almost all species tested, including Bacteroides fragilis at < or = 0.39 micrograms/mL. Although the other quinolones tested were active against gram-positive anaerobes, inhibiting their growth at < or = 1.56 micrograms/mL, these agents were less active against the B. fragilis group and Prevotella bivia (90% of which were inhibited at > or = 6.25 micrograms/mL). Mobiluncus species and G. vaginalis, which are well associated with bacterial vaginosis, were inhibited by DU-6859a at 0.1 microgram/mL. These results suggest that DU-6859a is a promising oral agent for the treatment of bacterial infections due to anaerobic bacteria; however, further studies, including determination of vaginal levels of this compound, should be performed to study the role of DU-6859a in the treatment of bacterial vaginosis.

Publication types

  • Comparative Study
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Administration, Oral
  • Anti-Infective Agents / administration & dosage
  • Anti-Infective Agents / pharmacology*
  • Bacteria, Anaerobic / drug effects*
  • Bacteria, Anaerobic / isolation & purification
  • Bacterial Infections / drug therapy
  • Bacteroides Infections / drug therapy
  • Bacteroides fragilis / drug effects
  • Bacteroides fragilis / isolation & purification
  • Female
  • Fluoroquinolones*
  • Gardnerella vaginalis / drug effects
  • Gardnerella vaginalis / isolation & purification
  • Humans
  • In Vitro Techniques
  • Japan
  • Microbial Sensitivity Tests
  • Quinolones / administration & dosage
  • Quinolones / pharmacology*
  • Vaginosis, Bacterial / drug therapy

Substances

  • Anti-Infective Agents
  • Fluoroquinolones
  • Quinolones
  • sitafloxacin