Adaptation of single cardiac ryanodine receptor channels

Biophys J. 1997 Feb;72(2 Pt 1):691-7. doi: 10.1016/s0006-3495(97)78705-8.

Abstract

Single cardiac ryanodine receptor (RyR) channel adaptation was previously defined with Ca2+ stimuli produced by flash photolysis of DM-nitrophen (caged-Ca+2). Photolysis of DM-nitrophen induced a very fast Ca+2 overshoot (Ca+2 spike) at the leading edge of the Ca+2 stimuli. It has been suggested that adaptation (tau approximately 1.3 s) may reflect Ca+2 slowly coming off the RyR Ca+2 activation sites following the faster Ca+2 spike (tau approximately 1 ms). This concern was addressed by defining the Ca2+ deactivation kinetics of single RyR channels in response to a rapid reduction in free Ca2+ concentration ([Ca2+]FREE). The [Ca2+]FREE was lowered by photolysis of Diazo-2. Single RyR channels deactivated (tau approximately 5.3 ms) quickly in response to the photolytically induced [Ca2+]FREE reduction. Improved estimates of the Ca2+ spike time course indicate that the Ca2+ spike is considerably faster (10-100-fold) than previously thought. Our data suggest that single RyRs are not significantly activated by fast Ca2+ spikes and that RyR adaptation is not due to deactivation following the fast Ca2+ spike. Thus, RyR adaptation may have an important impact on Ca2+ signaling in heart.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Acetates
  • Animals
  • Calcium / metabolism*
  • Calcium / pharmacology
  • Calcium Channels / metabolism*
  • Chelating Agents
  • Diazonium Compounds
  • Dogs
  • Ethylenediamines
  • In Vitro Techniques
  • Kinetics
  • Lipid Bilayers / metabolism
  • Muscle Proteins / metabolism*
  • Myocardium / metabolism*
  • Patch-Clamp Techniques
  • Phenoxyacetates
  • Phospholipids / metabolism
  • Photolysis
  • Ryanodine Receptor Calcium Release Channel
  • Sarcoplasmic Reticulum / metabolism*
  • Signal Transduction

Substances

  • Acetates
  • Calcium Channels
  • Chelating Agents
  • Diazonium Compounds
  • Ethylenediamines
  • Lipid Bilayers
  • Muscle Proteins
  • Phenoxyacetates
  • Phospholipids
  • Ryanodine Receptor Calcium Release Channel
  • diazo-2
  • DM-nitrophen
  • Calcium