Myb binding sites within the N-ras promoter repress transcription

Oncogene. 1997 Jul 10;15(2):193-202. doi: 10.1038/sj.onc.1201173.

Abstract

In vitro and in vivo methods were combined to determine the function of the three Myb binding sites (NrasI, NrasII and NrasIII) within the promoter region of the mouse N-ras gene. We found that the c-Myb DNA-binding domain can bind with high affinity to NrasI and NrasII, but with a reduced affinity to NrasIII. In contrast, the full length v-Myb protein from BM2 cells only bound to the middle one of the three sites, NrasII. Both c-Myb and v-Myb functioned as repressors and reduce the basal activity of the N-ras promoter by 60%, as determined by transient transfection experiments using different regions of the N-ras promoter. This repression required a functional Myb DNA-binding domain and could not be overcome by fusion to the potent VP16 activation domain. In electrophoretic mobility shift assays, the v-Myb protein is shown to be present in different conformations depending on its binding to the NrasII or the mim-1A site. The v-Myb conformation is thus suggested to play a critical role in the regulation of v-Myb activity.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Animals
  • Base Sequence
  • Binding Sites
  • Cells, Cultured
  • Chickens
  • Genes, ras*
  • Molecular Sequence Data
  • Promoter Regions, Genetic*
  • Protein Conformation
  • Proto-Oncogene Proteins / physiology*
  • Proto-Oncogene Proteins c-myb
  • Repressor Proteins / physiology*
  • Trans-Activators / physiology*
  • Transfection

Substances

  • Proto-Oncogene Proteins
  • Proto-Oncogene Proteins c-myb
  • Repressor Proteins
  • Trans-Activators