Abstract
The effect of NMDA receptor antagonist phencyclidine (PCP) on expression of cyclooxygenase (COX)-2 mRNA in the rat brain was studied. Administration of PCP (12.5, 25 or 50 mg/kg, i.p., 6 h) caused marked induction of COX-2 mRNA and heat shock gene hsp-70 mRNA, a marker of neuronal injury, in the retrosplenial cortex, in a dose-dependent manner. These results suggest that COX-2 may play a role in the neurotoxicity of NMDA receptor antagonists.
Publication types
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Research Support, Non-U.S. Gov't
MeSH terms
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Animals
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Brain Chemistry / drug effects
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Cerebral Cortex / chemistry
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Cerebral Cortex / enzymology*
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Cyclooxygenase 2
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Excitatory Amino Acid Antagonists / pharmacology*
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Female
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Gene Expression Regulation, Enzymologic / drug effects
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HSP70 Heat-Shock Proteins / genetics
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In Situ Hybridization
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Isoenzymes / genetics*
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Peroxidases / genetics
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Phencyclidine / pharmacology*
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Prostaglandin-Endoperoxide Synthases / genetics*
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RNA, Messenger / metabolism
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Rats
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Rats, Sprague-Dawley
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Receptors, N-Methyl-D-Aspartate / antagonists & inhibitors
Substances
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Excitatory Amino Acid Antagonists
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HSP70 Heat-Shock Proteins
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Isoenzymes
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RNA, Messenger
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Receptors, N-Methyl-D-Aspartate
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Peroxidases
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Cyclooxygenase 2
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Prostaglandin-Endoperoxide Synthases
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Phencyclidine