Activation of pyruvate dehydrogenase improves heart function and metabolism after hemorrhagic shock

J Mol Cell Cardiol. 1997 Sep;29(9):2465-74. doi: 10.1006/jmcc.1997.0483.

Abstract

This study was designed to test the hypothesis that activation of myocardial pyruvate dehydrogenase (PDH) would improve recovery of heart function after brief, severe hemorrhagic shock. Pentobarbital-anesthetized rats were instrumented to monitor arterial blood pressure and right ventricular pressures. Rats were hemorrhaged via femoral artery to 25-30 mmHg mean arterial pressure (MAP) for 60 min, followed by retransfusion of shed blood with either 1.0 cc saline with no dichloroacetate (-DCA) or 1.0 cc saline containing 150 mg/kg sodium dichloroacetate (+DCA). Rats were observed for 3 h after retransfusion. Hearts were freeze-clamped in situ for analysis of adenosine triphosphate (ATP), creatine phosphate (CrP), lactate and pyruvate content as well as PDH activity (PDHa) and total PDH activity (PDHt). Three h after retransfusion, the rate pressure product (RPP=HRxPSP) was 23 000+/-2733 with no DCA treatment v 36 2769 mmHg/min with DCA treatment (P<0.05, ANOVA). Treatment with DCA also increased myocardial tissue content of high energy phosphates (ATP=10.1+/-1.1 and CrP=5.8+/-1.0 micromol/g weight-DCA, v 15.1+/-0.9 and 14.7+/-1.0 micromol/g dry weight+DCA, P<0.05, both measurements). DCA administration also significantly reduced myocardial lactate contents (14.6+/-2.7 micromol/g dry weight-DCA v 5.9+/-1.0+DCA). Hemorrhagic shock did not change PDHa or PDHt compared to hearts obtained during the pre-hemorrhage period. Retransfusion with DCA significantly increased PDHa activity (6.8+/-1.1 micromol/g dry weight/min-DCA v 29.7+/-2.0 micromol/g dry weight/min+DCA). PDHt was not different between controls and DCA-treated groups. These data indicate that activation of myocardial PDH by adding DCA to retransfused blood improved heart function and metabolism after severe hemorrhagic shock.

Publication types

  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Adenosine Triphosphate / metabolism
  • Animals
  • Arteries
  • Blood Chemical Analysis
  • Blood Pressure
  • Dichloroacetic Acid / pharmacology*
  • Energy Metabolism
  • Heart / drug effects
  • Heart / physiology*
  • Hemodynamics
  • Lactic Acid / metabolism
  • Male
  • Myocardium / metabolism
  • Phosphates
  • Pyruvate Dehydrogenase Complex / drug effects
  • Pyruvate Dehydrogenase Complex / metabolism*
  • Pyruvic Acid / metabolism
  • Rats
  • Rats, Sprague-Dawley
  • Resuscitation
  • Shock, Hemorrhagic / drug therapy
  • Shock, Hemorrhagic / metabolism*
  • Ventricular Function

Substances

  • Phosphates
  • Pyruvate Dehydrogenase Complex
  • Lactic Acid
  • Pyruvic Acid
  • Adenosine Triphosphate
  • Dichloroacetic Acid