Electroretinogram in sucrose-fed diabetic rats treated with an aldose reductase inhibitor or an anticoagulant

Am J Physiol. 1997 Nov;273(5):E965-71. doi: 10.1152/ajpendo.1997.273.5.E965.

Abstract

To investigate the role of increased polyol pathway activity and hemodynamic deficits in the pathogenesis of diabetic retinopathy in non-insulin-dependent diabetes mellitus (NIDDM), Otsuka Long-Evans Tokushima fatty (OLETF) rats, an animal model of human NIDDM, were given water with or without 30% sucrose and some of them were fed laboratory chow containing 0.03% cilostazol, an anticoagulant, or 0.05% [5-(3-thienyl)tetrazol-1-yl] acetic acid monohydrate (TAT), an aldose reductase inhibitor, for 8 wk. Long-Evans Tokushima Otsuka (LETO) rats were used as nondiabetic controls. The peak latencies of oscillatory potentials of the electroretinogram in sucrose-fed OLETF rats were significantly prolonged compared with those in OLETF rats without sucrose feeding and LETO rats. There was a marked increase in platelet aggregability and a significant decrease in erythrocyte 2,3-diphosphoglycerate in sucrose-fed OLETF rats. Cilostazol significantly improved these parameters without changes in retinal levels of sorbitol and fructose. TAT, however, ameliorated all of these parameters. These findings confirm that the sucrose-fed OLETF rat is a useful animal model of retinopathy in human NIDDM and suggest that cilostazol improved diabetic retinopathy by modifying vascular factors, not by altering polyol pathway activity.

MeSH terms

  • 2,3-Diphosphoglycerate / metabolism
  • Aldehyde Reductase / antagonists & inhibitors*
  • Animals
  • Anticoagulants / pharmacology*
  • Blood Glucose / drug effects
  • Blood Glucose / metabolism
  • Body Weight / drug effects
  • Cilostazol
  • Diabetes Mellitus, Experimental / physiopathology*
  • Diabetes Mellitus, Type 2 / physiopathology*
  • Diabetic Retinopathy / physiopathology*
  • Dietary Sucrose / pharmacology*
  • Electroretinography / drug effects*
  • Enzyme Inhibitors / pharmacology*
  • Fructose / metabolism
  • Humans
  • Insulin / blood
  • Male
  • Platelet Aggregation / drug effects
  • Platelet Aggregation Inhibitors / pharmacology
  • Rats
  • Rats, Inbred Strains
  • Retina / drug effects
  • Retina / metabolism
  • Sorbitol / metabolism
  • Tetrazoles / pharmacology*
  • Thiophenes / pharmacology*
  • Triglycerides / blood

Substances

  • Anticoagulants
  • Blood Glucose
  • Dietary Sucrose
  • Enzyme Inhibitors
  • Insulin
  • Platelet Aggregation Inhibitors
  • Tetrazoles
  • Thiophenes
  • Triglycerides
  • (5-(3-thienyl)tetrazol-1-yl)acetic acid
  • 2,3-Diphosphoglycerate
  • Fructose
  • Sorbitol
  • Aldehyde Reductase
  • Cilostazol