Flavonoids reduce morphine withdrawal in-vitro

J Pharm Pharmacol. 1998 May;50(5):561-4. doi: 10.1111/j.2042-7158.1998.tb06199.x.

Abstract

The effects of quercetin, flavone, catechin and chrysin on the naloxone-precipitated withdrawal contracture of the acute morphine-dependent guinea-pig ileum have been investigated in-vitro. After 4 min in-vitro exposure to morphine a strong contracture of guinea-pig isolated ileum was observed after the addition of naloxone. All the flavonoids, injected 10 min before morphine at concentrations between 10(-7) and 10(-5) M, were capable of blocking naloxone-induced contracture after exposure to morphine in a concentration-dependent fashion. IC50 values calculated for quercetin, flavone, catechin and chrysin were 2.7 x 10(-6), 7.3 x 10(-7), 8.5 x 10(-7) and 5.3 x 10(-6) M, respectively. These results suggest that flavonoids might play an important role in the control of morphine withdrawal.

Publication types

  • Comparative Study

MeSH terms

  • Acetylcholine / pharmacology
  • Animals
  • Catechin / therapeutic use
  • Drug Interactions
  • Electric Stimulation
  • Flavonoids / therapeutic use*
  • Guinea Pigs
  • Ileum / drug effects
  • Male
  • Morphine / adverse effects*
  • Muscle Contraction / drug effects*
  • Naloxone / therapeutic use
  • Narcotic Antagonists / therapeutic use
  • Quercetin / therapeutic use
  • Substance Withdrawal Syndrome / drug therapy*

Substances

  • Flavonoids
  • Narcotic Antagonists
  • Naloxone
  • Morphine
  • Catechin
  • Quercetin
  • Acetylcholine