An essential methionine residue involved in substrate binding by phosphofructokinases

Biochem Biophys Res Commun. 1998 Sep 18;250(2):466-8. doi: 10.1006/bbrc.1998.9311.

Abstract

An alignment of all PPi-dependent phosphofructokinases and all allosteric ATP-dependent PFKs shows relatively few residues that are fully conserved. One residue that is conserved is a methionine residue that appears from the crystal structure of Escherichia coli PFK to be interacting with fructose 6-P. Very conservative substitutions for this methionine with leucine or isoleucine by site-directed mutagenesis of E. coli ATP-PFK and Entamoeba histolytica PPi-PFK produced profound decreases either in the apparent affinity for fructose 6-P or in maximal velocity, or both. Methionine provides a highly specific interaction with fructose 6-P for binding and for transition state stabilization.

Publication types

  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Allosteric Regulation
  • Animals
  • Binding Sites
  • Conserved Sequence
  • Entamoeba / enzymology*
  • Escherichia coli / enzymology*
  • Methionine
  • Mutation
  • Phosphofructokinase-1 / chemistry
  • Phosphofructokinase-1 / genetics*
  • Phosphofructokinase-1 / metabolism*
  • Substrate Specificity

Substances

  • Methionine
  • Phosphofructokinase-1