Non-fatal clozapine (LEPONEX) intoxication with toxicokinetic evaluation

Vet Hum Toxicol. 1999 Feb;41(1):20-2.

Abstract

A 29-y-old male attempted suicide with 3000 mg clozapine, 150 mg zopiclone, alprazolam and unknown quantities of alcohol. He was admitted in a deep hypotonic coma with respiratory depression, inhalation pneumonia and vascular collapse. Symptomatic treatment involved mechanical ventilation, vascular filling and antibiotics. The patient was discharged from the Intensive Care Unit 72 h after the suicide attempt with no sequelae. To detect and quantify clozapine in plasma, high-pressure liquid chromatography showed a 4 h absorption phase and a peak serum concentration of 5200 ng/ml. Three successive elimination t1/2 values of 38, 24 and 13 h were calculated.

Publication types

  • Case Reports

MeSH terms

  • Adult
  • Antipsychotic Agents / pharmacokinetics
  • Antipsychotic Agents / poisoning*
  • Chromatography, High Pressure Liquid
  • Clozapine / pharmacokinetics
  • Clozapine / poisoning*
  • Dose-Response Relationship, Drug
  • Evaluation Studies as Topic
  • Humans
  • Male
  • Schizophrenia / drug therapy*
  • Schizophrenia / metabolism
  • Treatment Outcome

Substances

  • Antipsychotic Agents
  • Clozapine