In vivo iron mobilisation evaluation of hydroxypyridinones in 59Fe-ferritin-loaded rat model

Biochem Pharmacol. 1999 Mar 1;57(5):559-66. doi: 10.1016/s0006-2952(98)00319-0.

Abstract

Although there are a number of well-characterised animal models available for testing and comparing the efficacy of iron chelators, most are expensive to operate and are not capable of providing rapid and reproducible results. The method described herein is based on the labelling of rat liver with 59Fe using rat 59Fe-ferritin. This method produces highly reproducible data of the type necessary for dose-response investigations, comparison of the efficacies of different administration routes, and structure activity studies.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Ferritins / metabolism*
  • Iron / metabolism*
  • Iron Chelating Agents / pharmacology*
  • Iron Radioisotopes / pharmacokinetics
  • Kinetics
  • Liver / metabolism*
  • Male
  • Models, Biological
  • Pyridones / chemistry
  • Pyridones / pharmacology*
  • Rats
  • Structure-Activity Relationship
  • Tissue Distribution

Substances

  • Iron Chelating Agents
  • Iron Radioisotopes
  • Pyridones
  • Ferritins
  • Iron