Walker KA - Search Results

1

Crystal structures of MMP-1 and -13 reveal the structural basis for selectivity of collagenase inhibitors.

Lovejoy B, Welch AR, Carr S, Luong C, Broka C, Hendricks RT, Campbell JA, Walker KA, Martin R, Van Wart H, Browner MF. Lovejoy B, et al. Among authors: walker ka. Nat Struct Biol. 1999 Mar;6(3):217-21. doi: 10.1038/6657. Nat Struct Biol. 1999. PMID: 10074939

2

Amino acid derived sulfonamide hydroxamates as inhibitors of procollagen C-proteinase. Part 2: Solid-phase optimization of side chains.

Dankwardt SM, Abbot SC, Broka CA, Martin RL, Chan CS, Springman EB, Van Wart HE, Walker KA. Dankwardt SM, et al. Among authors: walker ka. Bioorg Med Chem Lett. 2002 Apr 22;12(8):1233-5. doi: 10.1016/s0960-894x(02)00117-8. Bioorg Med Chem Lett. 2002. PMID: 11934595

3

Solid-phase synthesis of di- and tripeptidic hydroxamic acids as inhibitors of procollagen C-proteinase.

Dankwardt SM, Billedeau RJ, Lawley LK, Abbot SC, Martin RL, Chan CS, Van Wart HE, Walker KA. Dankwardt SM, et al. Among authors: walker ka. Bioorg Med Chem Lett. 2000 Nov 20;10(22):2513-6. doi: 10.1016/s0960-894x(00)00525-4. Bioorg Med Chem Lett. 2000. PMID: 11086718

4

Amino acid derived sulfonamide hydroxamates as inhibitors of procollagen C-proteinase: solid-phase synthesis of ornithine analogues.

Dankwardt SM, Martin RL, Chan CS, Van Wart HE, Walker KA, Delaet NG, Robinson LA. Dankwardt SM, et al. Among authors: walker ka. Bioorg Med Chem Lett. 2001 Aug 20;11(16):2085-8. doi: 10.1016/s0960-894x(01)00384-5. Bioorg Med Chem Lett. 2001. PMID: 11514144

5

Design and synthesis of orally active inhibitors of TNF synthesis as anti-rheumatoid arthritis drugs.

Chen JJ, Dewdney N, Lin X, Martin RL, Walker KA, Huang J, Chu F, Eugui E, Mirkovich A, Kim Y, Sarma K, Arzeno H, Van Wart HE. Chen JJ, et al. Among authors: walker ka. Bioorg Med Chem Lett. 2003 Nov 17;13(22):3951-4. doi: 10.1016/j.bmcl.2003.08.076. Bioorg Med Chem Lett. 2003. PMID: 14592482

6

Rational design of 6-methylsulfonylindoles as selective cyclooxygenase-2 inhibitors.

Campbell JA, Bordunov V, Broka CA, Browner MF, Kress JM, Mirzadegan T, Ramesha C, Sanpablo BF, Stabler R, Takahara P, Villasenor A, Walker KA, Wang JH, Welch M, Weller P. Campbell JA, et al. Among authors: walker ka. Bioorg Med Chem Lett. 2004 Sep 20;14(18):4741-5. doi: 10.1016/j.bmcl.2004.06.075. Bioorg Med Chem Lett. 2004. PMID: 15324899

7

Novel inhibitors of procollagen C-proteinase. Part 2: glutamic acid hydroxamates.

Robinson LA, Wilson DM, Delaet NG, Bradley EK, Dankwardt SM, Campbell JA, Martin RL, Van Wart HE, Walker KA, Sullivan RW. Robinson LA, et al. Among authors: walker ka. Bioorg Med Chem Lett. 2003 Jul 21;13(14):2381-4. doi: 10.1016/s0960-894x(03)00402-5. Bioorg Med Chem Lett. 2003. PMID: 12824039

8

Novel inhibitors of procollagen C-terminal proteinase. Part 1: diamino Acid hydroxamates.

Delaet NG, Robinson LA, Wilson DM, Sullivan RW, Bradley EK, Dankwardt SM, Martin RL, Van Wart HE, Walker KA. Delaet NG, et al. Among authors: walker ka. Bioorg Med Chem Lett. 2003 Jul 7;13(13):2101-4. doi: 10.1016/s0960-894x(03)00404-9. Bioorg Med Chem Lett. 2003. PMID: 12798313

9

Lactams as EP4 prostanoid receptor agonists. 3. Discovery of N-ethylbenzoic acid 2-pyrrolidinones as subtype selective agents.

Elworthy TR, Brill ER, Chiou SS, Chu F, Harris JR, Hendricks RT, Huang J, Kim W, Lach LK, Mirzadegan T, Yee C, Walker KA. Elworthy TR, et al. Among authors: walker ka. J Med Chem. 2004 Dec 2;47(25):6124-7. doi: 10.1021/jm049290a. J Med Chem. 2004. PMID: 15566283

10

Highly potent, non-basic 5-HT6 ligands. Site mutagenesis evidence for a second binding mode at 5-HT6 for antagonism.

Harris RN 3rd, Stabler RS, Repke DB, Kress JM, Walker KA, Martin RS, Brothers JM, Ilnicka M, Lee SW, Mirzadegan T. Harris RN 3rd, et al. Among authors: walker ka. Bioorg Med Chem Lett. 2010 Jun 1;20(11):3436-40. doi: 10.1016/j.bmcl.2010.03.110. Epub 2010 Apr 1. Bioorg Med Chem Lett. 2010. PMID: 20434910

Save citations to file

Email citations

Send citations to clipboard

Add to Collections

Add to My Bibliography

Create a file for external citation management software

Your saved search

Your RSS Feed

My Custom Filters

Publication date

Text availability

Article attribute

Article type

Article Language

Species

Sex

Age

Other

307 results

Search Page

Filters