Malamas M - Search Results

1

Prodrugs of CL316243: a selective beta3-adrenergic receptor agonist for treating obesity and diabetes.

Sum FW, Gilbert A, Venkatesan AM, Lim K, Wong V, O'Dell M, Francisco G, Chen Z, Grosu G, Baker J, Ellingboe J, Malamas M, Gunawan I, Primeau J, Largis E, Steiner K. Sum FW, et al. Among authors: malamas m. Bioorg Med Chem Lett. 1999 Jul 19;9(14):1921-6. doi: 10.1016/s0960-894x(99)00316-9. Bioorg Med Chem Lett. 1999. PMID: 10450954

2

2,4-Thiazolidinediones as potent and selective human beta3 agonists.

Hu B, Ellingboe J, Gunawan I, Han S, Largis E, Li Z, Malamas M, Mulvey R, Oliphant A, Sum FW, Tillett J, Wong V. Hu B, et al. Among authors: malamas m. Bioorg Med Chem Lett. 2001 Mar 26;11(6):757-60. doi: 10.1016/s0960-894x(01)00063-4. Bioorg Med Chem Lett. 2001. PMID: 11277513

3

New oxadiazolidinedione derivatives as potent and selective human beta3 agonists.

Hu B, Malamas M, Ellingboe J, Largis E, Han S, Mulvey R, Tillett J. Hu B, et al. Among authors: malamas m. Bioorg Med Chem Lett. 2001 Apr 23;11(8):981-4. doi: 10.1016/s0960-894x(01)00147-0. Bioorg Med Chem Lett. 2001. PMID: 11327605

4

Novel (4-piperidin-1-yl)-phenyl sulfonamides as potent and selective human beta(3) agonists.

Hu B, Ellingboe J, Han S, Largis E, Lim K, Malamas M, Mulvey R, Niu C, Oliphant A, Pelletier J, Singanallore T, Sum FW, Tillett J, Wong V. Hu B, et al. Among authors: malamas m. Bioorg Med Chem. 2001 Aug;9(8):2045-59. doi: 10.1016/s0968-0896(01)00114-6. Bioorg Med Chem. 2001. PMID: 11504641

5

New azolidinediones as inhibitors of protein tyrosine phosphatase 1B with antihyperglycemic properties.

Malamas MS, Sredy J, Gunawan I, Mihan B, Sawicki DR, Seestaller L, Sullivan D, Flam BR. Malamas MS, et al. J Med Chem. 2000 Mar 9;43(5):995-1010. doi: 10.1021/jm990476x. J Med Chem. 2000. PMID: 10715163

6

Antihyperglycemic activity of new 1,2,4-oxadiazolidine-3,5-diones.

Malamas MS, Sredy J, McCaleb M, Gunawan I, Mihan B, Sullivan D. Malamas MS, et al. Eur J Med Chem. 2001 Jan;36(1):31-42. doi: 10.1016/s0223-5234(00)01191-0. Eur J Med Chem. 2001. PMID: 11231047

7

Design and synthesis of aryl diphenolic azoles as potent and selective estrogen receptor-beta ligands.

Malamas MS, Manas ES, McDevitt RE, Gunawan I, Xu ZB, Collini MD, Miller CP, Dinh T, Henderson RA, Keith JC Jr, Harris HA. Malamas MS, et al. J Med Chem. 2004 Oct 7;47(21):5021-40. doi: 10.1021/jm049719y. J Med Chem. 2004. PMID: 15456246

8

Azole phenoxy hydroxyureas as selective and orally active inhibitors of 5-lipoxygenase.

Malamas MS, Carlson RP, Grimes D, Howell R, Glaser K, Gunawan I, Nelson JA, Kanzelberger M, Shah U, Hartman DA. Malamas MS, et al. J Med Chem. 1996 Jan 5;39(1):237-45. doi: 10.1021/jm950363n. J Med Chem. 1996. PMID: 8568813

9

Acylguanidine inhibitors of beta-secretase: optimization of the pyrrole ring substituents extending into the S1' substrate binding pocket.

Jennings LD, Cole DC, Stock JR, Sukhdeo MN, Ellingboe JW, Cowling R, Jin G, Manas ES, Fan KY, Malamas MS, Harrison BL, Jacobsen S, Chopra R, Lohse PA, Moore WJ, O'Donnell MM, Hu Y, Robichaud AJ, Turner MJ, Wagner E, Bard J. Jennings LD, et al. Among authors: malamas ms. Bioorg Med Chem Lett. 2008 Jan 15;18(2):767-71. doi: 10.1016/j.bmcl.2007.11.043. Epub 2007 Nov 17. Bioorg Med Chem Lett. 2008. PMID: 18068983

10

Acylguanidine inhibitors of beta-secretase: optimization of the pyrrole ring substituents extending into the S1 and S3 substrate binding pockets.

Cole DC, Stock JR, Chopra R, Cowling R, Ellingboe JW, Fan KY, Harrison BL, Hu Y, Jacobsen S, Jennings LD, Jin G, Lohse PA, Malamas MS, Manas ES, Moore WJ, O'Donnell MM, Olland AM, Robichaud AJ, Svenson K, Wu J, Wagner E, Bard J. Cole DC, et al. Among authors: malamas ms. Bioorg Med Chem Lett. 2008 Feb 1;18(3):1063-6. doi: 10.1016/j.bmcl.2007.12.010. Epub 2007 Dec 10. Bioorg Med Chem Lett. 2008. PMID: 18162398

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