Millet R - Search Results

1

Conformation of the tripeptide Cbz-Pro-Leu-Trp-OBzl(CF3)2 deduced from two-dimensional 1H-NMR and conformational energy calculations is related to its affinity for NK1-receptor.

Millet R, Goossens L, Goossens JF, Chavatte P, Bertrand-Caumont K, Houssin R, Hénichart JP. Millet R, et al. J Pept Sci. 2001 Jun;7(6):323-30. doi: 10.1002/psc.326. J Pept Sci. 2001. PMID: 11461046

2

A flexible approach to the design of new potent substance P receptor ligands.

Millet R, Goossens L, Bertrand-Caumont K, Goossens JF, Houssin R, Hénichart JP. Millet R, et al. J Pharm Pharmacol. 2001 Jul;53(7):929-34. doi: 10.1211/0022357011776324. J Pharm Pharmacol. 2001. PMID: 11480541

3

Novel potent substance P and neurokinin A receptor antagonists. Conception, synthesis and biological evaluation of indolizine derivatives.

Millet R, Domarkas J, Rigo B, Goossens L, Goossens JF, Houssin R, Hénichart JP. Millet R, et al. Bioorg Med Chem. 2002 Sep;10(9):2905-12. doi: 10.1016/s0968-0896(02)00144-x. Bioorg Med Chem. 2002. PMID: 12110311

4

Potent and selective farnesyl transferase inhibitors.

Millet R, Domarkas J, Houssin R, Gilleron P, Goossens JF, Chavatte P, Logé C, Pommery N, Pommery J, Hénichart JP. Millet R, et al. J Med Chem. 2004 Dec 30;47(27):6812-20. doi: 10.1021/jm030502y. J Med Chem. 2004. PMID: 15615530

5

Synthesis of a novel conformationally restricted Val-Phe dipeptidomimetic.

Gilleron P, Millet R, Domarkas J, Farce A, Houssin R, Hénichart JP. Gilleron P, et al. Among authors: millet r. J Pept Sci. 2006 Feb;12(2):140-6. doi: 10.1002/psc.688. J Pept Sci. 2006. PMID: 15948143

6

Novel N-(4-Piperidinyl)benzamide antimalarials with mammalian protein farnesyltransferase inhibitory activity.

Ryckebusch A, Gilleron P, Millet R, Houssin R, Lemoine A, Pommery N, Grellier P, Sergheraert C, Hénichart JP. Ryckebusch A, et al. Among authors: millet r. Chem Pharm Bull (Tokyo). 2005 Oct;53(10):1324-6. doi: 10.1248/cpb.53.1324. Chem Pharm Bull (Tokyo). 2005. PMID: 16204993 Free article.

7

Novel 4-oxo-1,4-dihydroquinoline-3-carboxamide derivatives as new CB2 cannabinoid receptors agonists: synthesis, pharmacological properties and molecular modeling.

Stern E, Muccioli GG, Millet R, Goossens JF, Farce A, Chavatte P, Poupaert JH, Lambert DM, Depreux P, Hénichart JP. Stern E, et al. Among authors: millet r. J Med Chem. 2006 Jan 12;49(1):70-9. doi: 10.1021/jm050467q. J Med Chem. 2006. PMID: 16392793

8

Solid-phase synthesis and pharmacological evaluation of a library of peptidomimetics as potential farnesyltransferase inhibitors: an approach to new lead compounds.

Gilleron P, Millet R, Houssin R, Wlodarczyk N, Farce A, Lemoine A, Goossens JF, Chavatte P, Pommery N, Hénichart JP. Gilleron P, et al. Among authors: millet r. Eur J Med Chem. 2006 Jun;41(6):745-55. doi: 10.1016/j.ejmech.2006.03.017. Epub 2006 May 2. Eur J Med Chem. 2006. PMID: 16647166

9

In vitro and in vivo evaluation of two rational-designed nonpeptidic farnesyltransferase inhibitors on HT29 human colon cancer cell lines.

Wlodarczyk N, Gilleron P, Millet R, Houssin R, Goossens JF, Lemoine A, Pommery N, Wei MX, Hénichart JP. Wlodarczyk N, et al. Among authors: millet r. Oncol Res. 2005;16(3):107-18. doi: 10.3727/000000006783981170. Oncol Res. 2005. PMID: 16925112

10

Design, synthesis and biological evaluation of substituted dioxodibenzothiazepines and dibenzocycloheptanes as farnesyltransferase inhibitors.

Gilleron P, Wlodarczyk N, Houssin R, Farce A, Laconde G, Goossens JF, Lemoine A, Pommery N, Hénichart JP, Millet R. Gilleron P, et al. Among authors: millet r. Bioorg Med Chem Lett. 2007 Oct 1;17(19):5465-71. doi: 10.1016/j.bmcl.2007.07.002. Epub 2007 Jul 7. Bioorg Med Chem Lett. 2007. PMID: 17827015

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