Chiral N,N-disubstituted trifluoro-3-amino-2-propanols are potent inhibitors of cholesteryl ester transfer protein.
Durley RC, Grapperhaus ML, Hickory BS, Massa MA, Wang JL, Spangler DP, Mischke DA, Parnas BL, Fobian YM, Rath NP, Honda DD, Zeng M, Connolly DT, Heuvelman DM, Witherbee BJ, Melton MA, Glenn KC, Krul ES, Smith ME, Sikorski JA.
Durley RC, et al. Among authors: zeng m.
J Med Chem. 2002 Aug 29;45(18):3891-904. doi: 10.1021/jm020038h.
J Med Chem. 2002.
PMID: 12190312