Sim E - Search Results

1

An approach to identifying novel substrates of bacterial arylamine N-acetyltransferases.

Brooke EW, Davies SG, Mulvaney AW, Pompeo F, Sim E, Vickers RJ. Brooke EW, et al. Among authors: sim e. Bioorg Med Chem. 2003 Apr 3;11(7):1227-34. doi: 10.1016/s0968-0896(02)00642-9. Bioorg Med Chem. 2003. PMID: 12628650

2

Expression and purification of the rifamycin amide synthase, RifF, an enzyme homologous to the prokaryotic arylamine N-acetyltransferases.

Pompeo F, Mushtaq A, Sim E. Pompeo F, et al. Among authors: sim e. Protein Expr Purif. 2002 Feb;24(1):138-51. doi: 10.1006/prep.2001.1550. Protein Expr Purif. 2002. PMID: 11812235

3

The pharmacogenetics of NAT: structural aspects.

Pompeo F, Brooke E, Kawamura A, Mushtaq A, Sim E. Pompeo F, et al. Among authors: sim e. Pharmacogenomics. 2002 Jan;3(1):19-30. doi: 10.1517/14622416.3.1.19. Pharmacogenomics. 2002. PMID: 11966400 Review.

4

Synthesis and in vitro evaluation of novel small molecule inhibitors of bacterial arylamine N-acetyltransferases (NATs).

Brooke EW, Davies SG, Mulvaney AW, Okada M, Pompeo F, Sim E, Vickers RJ, Westwood IM. Brooke EW, et al. Among authors: sim e. Bioorg Med Chem Lett. 2003 Aug 4;13(15):2527-30. doi: 10.1016/s0960-894x(03)00484-0. Bioorg Med Chem Lett. 2003. PMID: 12852958

5

Inhibition of mycobacterial arylamine N-acetyltransferase contributes to anti-mycobacterial activity of Warburgia salutaris.

Madikane VE, Bhakta S, Russell AJ, Campbell WE, Claridge TD, Elisha BG, Davies SG, Smith P, Sim E. Madikane VE, et al. Among authors: sim e. Bioorg Med Chem. 2007 May 15;15(10):3579-86. doi: 10.1016/j.bmc.2007.02.011. Epub 2007 Feb 11. Bioorg Med Chem. 2007. PMID: 17368035

6

Selective small molecule inhibitors of the potential breast cancer marker, human arylamine N-acetyltransferase 1, and its murine homologue, mouse arylamine N-acetyltransferase 2.

Russell AJ, Westwood IM, Crawford MH, Robinson J, Kawamura A, Redfield C, Laurieri N, Lowe ED, Davies SG, Sim E. Russell AJ, et al. Among authors: sim e. Bioorg Med Chem. 2009 Jan 15;17(2):905-18. doi: 10.1016/j.bmc.2008.11.032. Epub 2008 Nov 19. Bioorg Med Chem. 2009. PMID: 19059786

7

Novel small-molecule inhibitors of arylamine N-acetyltransferases: drug discovery by high-throughput screening.

Westwood IM, Kawamura A, Russell AJ, Sandy J, Davies SG, Sim E. Westwood IM, et al. Among authors: sim e. Comb Chem High Throughput Screen. 2011 Feb;14(2):117-24. doi: 10.2174/138620711794474051. Comb Chem High Throughput Screen. 2011. PMID: 21118080

8

Identification of arylamine N-acetyltransferase inhibitors as an approach towards novel anti-tuberculars.

Westwood IM, Bhakta S, Russell AJ, Fullam E, Anderton MC, Kawamura A, Mulvaney AW, Vickers RJ, Bhowruth V, Besra GS, Lalvani A, Davies SG, Sim E. Westwood IM, et al. Among authors: sim e. Protein Cell. 2010 Jan;1(1):82-95. doi: 10.1007/s13238-010-0006-1. Epub 2010 Mar 18. Protein Cell. 2010. PMID: 21204000 Free PMC article.

9

Design, synthesis and structure-activity relationships of 3,5-diaryl-1H-pyrazoles as inhibitors of arylamine N-acetyltransferase.

Fullam E, Talbot J, Abuhammed A, Westwood I, Davies SG, Russell AJ, Sim E. Fullam E, et al. Among authors: sim e. Bioorg Med Chem Lett. 2013 May 1;23(9):2759-64. doi: 10.1016/j.bmcl.2013.02.052. Epub 2013 Feb 22. Bioorg Med Chem Lett. 2013. PMID: 23518278

10

Structure and mechanism of arylamine N-acetyltransferases.

Westwood IM, Kawamura A, Fullam E, Russell AJ, Davies SG, Sim E. Westwood IM, et al. Among authors: sim e. Curr Top Med Chem. 2006;6(15):1641-54. doi: 10.2174/156802606778108979. Curr Top Med Chem. 2006. PMID: 16918475 Review.

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