Scilimati A - Search Results

1

Optimal requirements for high affinity and use-dependent block of skeletal muscle sodium channel by N-benzyl analogs of tocainide-like compounds.

De Luca A, Talon S, De Bellis M, Desaphy JF, Lentini G, Corbo F, Scilimati A, Franchini C, Tortorella V, Camerino DC. De Luca A, et al. Among authors: scilimati a. Mol Pharmacol. 2003 Oct;64(4):932-45. doi: 10.1124/mol.64.4.932. Mol Pharmacol. 2003. PMID: 14500750

2

Synthesis of new 2,6-prolylxylidide analogues of tocainide as stereoselective blockers of voltage-gated Na(+) channels with increased potency and improved use-dependent activity.

Franchini C, Corbo F, Lentini G, Bruno G, Scilimati A, Tortorella V, Conte Camerino D, De Luca A. Franchini C, et al. Among authors: scilimati a. J Med Chem. 2000 Oct 5;43(20):3792-8. doi: 10.1021/jm000931l. J Med Chem. 2000. PMID: 11020295

3

Increased rigidity of the chiral centre of tocainide favours stereoselectivity and use-dependent block of skeletal muscle Na(+) channels enhancing the antimyotonic activity in vivo.

Talon S, De Luca A, De Bellis M, Desaphy JF, Lentini G, Scilimati A, Corbo F, Franchini C, Tortorella P, Jockusch H, Conte Camerino D. Talon S, et al. Among authors: scilimati a. Br J Pharmacol. 2001 Dec;134(7):1523-31. doi: 10.1038/sj.bjp.0704366. Br J Pharmacol. 2001. PMID: 11724759 Free PMC article.

4

Optically active mexiletine analogues as stereoselective blockers of voltage-gated Na(+) channels.

Franchini C, Carocci A, Catalano A, Cavalluzzi MM, Corbo F, Lentini G, Scilimati A, Tortorella P, Camerino DC, De Luca A. Franchini C, et al. Among authors: scilimati a. J Med Chem. 2003 Nov 20;46(24):5238-48. doi: 10.1021/jm030865y. J Med Chem. 2003. PMID: 14613326

5

Synthesis and biological evaluation of new clofibrate analogues as potential PPARalpha agonists.

Perrone MG, Santandrea E, Dell'Uomo N, Giannessi F, Milazzo FM, Sciarroni AF, Scilimati A, Tortorella V. Perrone MG, et al. Among authors: scilimati a. Eur J Med Chem. 2005 Feb;40(2):143-54. doi: 10.1016/j.ejmech.2004.09.018. Eur J Med Chem. 2005. PMID: 15694649

6

Constrained analogues of tocainide as potent skeletal muscle sodium channel blockers towards the development of antimyotonic agents.

Catalano A, Carocci A, Corbo F, Franchini C, Muraglia M, Scilimati A, De Bellis M, De Luca A, Camerino DC, Sinicropi MS, Tortorella V. Catalano A, et al. Among authors: scilimati a. Eur J Med Chem. 2008 Nov;43(11):2535-40. doi: 10.1016/j.ejmech.2008.01.023. Epub 2008 Jan 31. Eur J Med Chem. 2008. PMID: 18342401

7

Myogenic effect of SP-1f and SP-1h two novel β3-adrenoceptor (β3-AR) agonists in human colonic circular smooth muscle.

Maselli MA, Trisolini P, Ignazzi A, Notarnicola M, Lorusso D, Pezzolla F, Iacobazzi D, Scilimati A, Perrone MG. Maselli MA, et al. Among authors: scilimati a. Eur J Pharmacol. 2014 Jan 15;723:62-6. doi: 10.1016/j.ejphar.2013.11.010. Epub 2013 Nov 22. Eur J Pharmacol. 2014. PMID: 24275352

8

Selective cyclooxygenase-1 inhibition by p6 and gastrotoxicity: preliminary investigation.

Perrone MG, Lofrumento DD, Vitale P, De Nuccio F, La Pesa V, Panella A, Calvello R, Cianciulli A, Panaro MA, Scilimati A. Perrone MG, et al. Among authors: scilimati a. Pharmacology. 2015;95(1-2):22-8. doi: 10.1159/000369826. Epub 2015 Jan 9. Pharmacology. 2015. PMID: 25591798

9

A novel injectable formulation of 6-fluoro-l-DOPA imaging agent for diagnosis of neuroendocrine tumors and Parkinson's disease.

Trapani A, Tricarico D, Mele A, Maqoud F, Mandracchia D, Vitale P, Capriati V, Trapani G, Dimiccoli V, Tolomeo A, Scilimati A. Trapani A, et al. Among authors: scilimati a. Int J Pharm. 2017 Mar 15;519(1-2):304-313. doi: 10.1016/j.ijpharm.2017.01.038. Epub 2017 Jan 21. Int J Pharm. 2017. PMID: 28119123

10

Novel synthesis of 3,4-diarylisoxazole analogues of valdecoxib: reversal cyclooxygenase-2 selectivity by sulfonamide group removal.

Di Nunno L, Vitale P, Scilimati A, Tacconelli S, Patrignani P. Di Nunno L, et al. Among authors: scilimati a. J Med Chem. 2004 Sep 23;47(20):4881-90. doi: 10.1021/jm040782x. J Med Chem. 2004. PMID: 15369392

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