Singer RA - Search Results

1

A general route to the synthesis of 1,5-methano- and 1,5-ethano- 2,3,4,5-tetrahydro-1H-3-benzazepines.

O'Donnell CJ, Singer RA, Brubaker JD, McKinley JD. O'Donnell CJ, et al. Among authors: singer ra. J Org Chem. 2004 Aug 20;69(17):5756-9. doi: 10.1021/jo049122q. J Org Chem. 2004. PMID: 15307752

2

Preparation of 1,5-methano-2,3,4,5- tetrahydro-1H-3-benzazepine via Pd-catalyzed cyclization.

Singer RA, McKinley JD, Barbe G, Farlow RA. Singer RA, et al. Org Lett. 2004 Jul 8;6(14):2357-60. doi: 10.1021/ol049316s. Org Lett. 2004. PMID: 15228278

3

Aminocarbonylation of aryl tosylates to carboxamides.

Chung S, Sach N, Choi C, Yang X, Drozda SE, Singer RA, Wright SW. Chung S, et al. Among authors: singer ra. Org Lett. 2015 Jun 5;17(11):2848-51. doi: 10.1021/acs.orglett.5b01283. Epub 2015 May 21. Org Lett. 2015. PMID: 25994500

4

Diastereoselective Diboration of Cyclic Alkenes: Application to the Synthesis of Aristeromycin.

Vendola AJ, Allais C, Dechert-Schmitt AR, Lee JT, Singer RA, Morken JP. Vendola AJ, et al. Among authors: singer ra. Org Lett. 2021 Apr 16;23(8):2863-2867. doi: 10.1021/acs.orglett.1c00353. Epub 2021 Apr 1. Org Lett. 2021. PMID: 33792325

5

Construction of Azacycles by Intramolecular Amination of Organoboronates and Organobis(boronates).

Xu P, Zhang M, Ingoglia B, Allais C, Dechert-Schmitt AR, Singer RA, Morken JP. Xu P, et al. Among authors: singer ra. Org Lett. 2021 May 7;23(9):3379-3383. doi: 10.1021/acs.orglett.1c00856. Epub 2021 Apr 14. Org Lett. 2021. PMID: 33852313

6

Early Clinical Development of Lufotrelvir as a Potential Therapy for COVID-19.

Allais C, Bernhardson D, Brown AR, Chinigo GM, Desrosiers JN, DiRico KJ, Hotham I, Jones BP, Kulkarni SA, Lewis CA, Lira R, Loach RP, Morse PD, Mousseau JJ, Perry MA, Peng Z, Place DW, Rane AM, Samp L, Singer RA, Wang Z, Weisenburger GA, Yayla HG, Zanghi JM. Allais C, et al. Among authors: singer ra. Org Process Res Dev. 2023 Feb 3:acs.oprd.2c00375. doi: 10.1021/acs.oprd.2c00375. Online ahead of print. Org Process Res Dev. 2023. PMID: 37552749 Review.

7

Distal Stereocontrol Using Guanidinylated Peptides as Multifunctional Ligands: Desymmetrization of Diarylmethanes via Ullman Cross-Coupling.

Kim B, Chinn AJ, Fandrick DR, Senanayake CH, Singer RA, Miller SJ. Kim B, et al. Among authors: singer ra. J Am Chem Soc. 2016 Jun 29;138(25):7939-45. doi: 10.1021/jacs.6b03444. Epub 2016 Jun 15. J Am Chem Soc. 2016. PMID: 27254785 Free PMC article.

8

Development of a targeted polymorph screening approach for a complex polymorphic and highly solvating API.

Campeta AM, Chekal BP, Abramov YA, Meenan PA, Henson MJ, Shi B, Singer RA, Horspool KR. Campeta AM, et al. Among authors: singer ra. J Pharm Sci. 2010 Sep;99(9):3874-86. doi: 10.1002/jps.22230. J Pharm Sci. 2010. PMID: 20575000

9

Stereocontrolled Pericyclic and Radical Cycloaddition Reactions of Readily Accessible Chiral Alkenyl Diazaborolidines.

Zhang M, Xu P, Vendola AJ, Allais C, Dechert Schmitt AM, Singer RA, Morken JP. Zhang M, et al. Among authors: singer ra. Angew Chem Int Ed Engl. 2022 Jul 25;61(30):e202205454. doi: 10.1002/anie.202205454. Epub 2022 Jun 8. Angew Chem Int Ed Engl. 2022. PMID: 35587213 Free PMC article.

10

Desymmetrization of Vicinal Bis(boronic) Esters by Enantioselective Suzuki-Miyaura Cross-Coupling Reaction.

Zhang M, Lee PS, Allais C, Singer RA, Morken JP. Zhang M, et al. Among authors: singer ra. J Am Chem Soc. 2023 Apr 6:10.1021/jacs.3c01571. doi: 10.1021/jacs.3c01571. Online ahead of print. J Am Chem Soc. 2023. PMID: 37023255 Free PMC article.

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