Schreiner E - Search Results

1

6-[2-(adamantylidene)-hydroxybenzoxazole]-O-sulfamate, a steroid sulfatase inhibitor for the treatment of androgen- and estrogen-dependent diseases.

Billich A, Meingassner JG, Nussbaumer P, Desrayaud S, Lam C, Winiski A, Schreiner E. Billich A, et al. Among authors: schreiner e. J Steroid Biochem Mol Biol. 2004 Sep;92(1-2):29-37. doi: 10.1016/j.jsbmb.2004.06.004. J Steroid Biochem Mol Biol. 2004. PMID: 15544928

2

6-(2-adamantan-2-ylidene-hydroxybenzoxazole)-O-sulfamate: a potent non-steroidal irreversible inhibitor of human steroid sulfatase.

Schreiner EP, Wolff B, Winiski AP, Billich A. Schreiner EP, et al. Bioorg Med Chem Lett. 2003 Dec 15;13(24):4313-6. doi: 10.1016/j.bmcl.2003.09.050. Bioorg Med Chem Lett. 2003. PMID: 14643316

3

Estrone formate: a novel type of irreversible inhibitor of human steroid sulfatase.

Schreiner EP, Billich A. Schreiner EP, et al. Bioorg Med Chem Lett. 2004 Oct 4;14(19):4999-5002. doi: 10.1016/j.bmcl.2004.07.013. Bioorg Med Chem Lett. 2004. PMID: 15341968

4

Inhibitors of HIV-1 proteinase containing 2-heterosubstituted 4-amino-3-hydroxy-5-phenylpentanoic acid: synthesis, enzyme inhibition, and antiviral activity.

Scholz D, Billich A, Charpiot B, Ettmayer P, Lehr P, Rosenwirth B, Schreiner E, Gstach H. Scholz D, et al. Among authors: schreiner e. J Med Chem. 1994 Sep 16;37(19):3079-89. doi: 10.1021/jm00045a013. J Med Chem. 1994. PMID: 7932531

5

Inhibition of vascular endothelial growth factor cotranslational translocation by the cyclopeptolide CAM741.

Harant H, Wolff B, Schreiner EP, Oberhauser B, Hofer L, Lettner N, Maier S, de Vries JE, Lindley IJ. Harant H, et al. Among authors: schreiner ep. Mol Pharmacol. 2007 Jun;71(6):1657-65. doi: 10.1124/mol.107.034249. Epub 2007 Mar 16. Mol Pharmacol. 2007. PMID: 17369307

6

Selective inhibition of cotranslational translocation of vascular cell adhesion molecule 1.

Besemer J, Harant H, Wang S, Oberhauser B, Marquardt K, Foster CA, Schreiner EP, de Vries JE, Dascher-Nadel C, Lindley IJ. Besemer J, et al. Among authors: schreiner ep. Nature. 2005 Jul 14;436(7048):290-3. doi: 10.1038/nature03670. Nature. 2005. PMID: 16015337

7

Synthesis of ether analogues derived from HUN-7293 and evaluation as inhibitors of VCAM-1 expression.

Schreiner EP, Kern M, Steck A, Foster CA. Schreiner EP, et al. Bioorg Med Chem Lett. 2004 Oct 4;14(19):5003-6. doi: 10.1016/j.bmcl.2004.07.012. Bioorg Med Chem Lett. 2004. PMID: 15341969

8

Leptomycin B inactivates CRM1/exportin 1 by covalent modification at a cysteine residue in the central conserved region.

Kudo N, Matsumori N, Taoka H, Fujiwara D, Schreiner EP, Wolff B, Yoshida M, Horinouchi S. Kudo N, et al. Among authors: schreiner ep. Proc Natl Acad Sci U S A. 1999 Aug 3;96(16):9112-7. doi: 10.1073/pnas.96.16.9112. Proc Natl Acad Sci U S A. 1999. PMID: 10430904 Free PMC article.

9

A convenient protocol for selective cleavage of 2-hydroxy acid amides. Application to semisynthesis of the cyclic heptapeptide aza HUN-7293.

Schreiner EP, Kern M, Steck A. Schreiner EP, et al. J Org Chem. 2002 Nov 29;67(24):8299-304. doi: 10.1021/jo025979g. J Org Chem. 2002. PMID: 12444606

10

Synthesis of enantiopure antiobesity drug lorcaserin.

Smilovic IG, Cluzeau J, Richter F, Nerdinger S, Schreiner E, Laus G, Schottenberger H. Smilovic IG, et al. Among authors: schreiner e. Bioorg Med Chem. 2018 May 15;26(9):2686-2690. doi: 10.1016/j.bmc.2018.02.038. Epub 2018 Feb 21. Bioorg Med Chem. 2018. PMID: 29496415

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