Whalley ET - Search Results

1

Synthesis of alkyne derivatives of a novel triazolopyrazine as A(2A) adenosine receptor antagonists.

Yao G, Haque S, Sha L, Kumaravel G, Wang J, Engber TM, Whalley ET, Conlon PR, Chang H, Kiesman WF, Petter RC. Yao G, et al. Among authors: whalley et. Bioorg Med Chem Lett. 2005 Feb 1;15(3):511-5. doi: 10.1016/j.bmcl.2004.11.062. Bioorg Med Chem Lett. 2005. PMID: 15664803

2

Novel bicyclic piperazine derivatives of triazolotriazine and triazolopyrimidines as highly potent and selective adenosine A2A receptor antagonists.

Peng H, Kumaravel G, Yao G, Sha L, Wang J, Van Vlijmen H, Bohnert T, Huang C, Vu CB, Ensinger CL, Chang H, Engber TM, Whalley ET, Petter RC. Peng H, et al. Among authors: whalley et. J Med Chem. 2004 Dec 2;47(25):6218-29. doi: 10.1021/jm0494321. J Med Chem. 2004. PMID: 15566292

3

Design, synthesis, and analysis of a polyethelene glycol-modified (PEGylated) small molecule inhibitor of integrin {alpha}4{beta}1 with improved pharmaceutical properties.

Pepinsky RB, Lee WC, Cornebise M, Gill A, Wortham K, Chen LL, Leone DR, Giza K, Dolinski BM, Perper S, Nickerson-Nutter C, Lepage D, Chakraborty A, Whalley ET, Petter RC, Adams SP, Lobb RR, Scott DM. Pepinsky RB, et al. Among authors: whalley et. J Pharmacol Exp Ther. 2005 Feb;312(2):742-50. doi: 10.1124/jpet.104.075648. Epub 2004 Oct 14. J Pharmacol Exp Ther. 2005. PMID: 15485895

4

Comparison of three different A1 adenosine receptor antagonists on infarct size and multiple cycle ischemic preconditioning in anesthetized dogs.

Auchampach JA, Jin X, Moore J, Wan TC, Kreckler LM, Ge ZD, Narayanan J, Whalley E, Kiesman W, Ticho B, Smits G, Gross GJ. Auchampach JA, et al. J Pharmacol Exp Ther. 2004 Mar;308(3):846-56. doi: 10.1124/jpet.103.057943. Epub 2003 Nov 21. J Pharmacol Exp Ther. 2004. PMID: 14634049

5

An assessment of the mechanistic differences between two integrin alpha 4 beta 1 inhibitors, the monoclonal antibody TA-2 and the small molecule BIO5192, in rat experimental autoimmune encephalomyelitis.

Leone DR, Giza K, Gill A, Dolinski BM, Yang W, Perper S, Scott DM, Lee WC, Cornebise M, Wortham K, Nickerson-Nutter C, Chen LL, LePage D, Spell JC, Whalley ET, Petter RC, Adams SP, Lobb RR, Pepinsky RB. Leone DR, et al. Among authors: whalley et. J Pharmacol Exp Ther. 2003 Jun;305(3):1150-62. doi: 10.1124/jpet.102.047332. Epub 2003 Mar 6. J Pharmacol Exp Ther. 2003. PMID: 12626659

6

Bradykinin receptor antagonists containing N-substituted amino acids: in vitro and in vivo B(2) and B(1) receptor antagonist activity.

Goodfellow VS, Marathe MV, Kuhlman KG, Fitzpatrick TD, Cuadrado D, Hanson W, Zuzack JS, Ross SE, Wieczorek M, Burkard M, Whalley ET. Goodfellow VS, et al. Among authors: whalley et. J Med Chem. 1996 Mar 29;39(7):1472-84. doi: 10.1021/jm950716i. J Med Chem. 1996. PMID: 8691478

7

Design, synthesis, and in vitro activity of bis(succinimido)hexane peptide heterodimers with combined B1 and B2 antagonist activity.

Cheronis JC, Whalley ET, Allen LG, Loy SD, Elder MW, Duggan MJ, Gross KL, Blodgett JK. Cheronis JC, et al. Among authors: whalley et. J Med Chem. 1994 Feb 4;37(3):348-55. doi: 10.1021/jm00029a006. J Med Chem. 1994. PMID: 8308862

8

Dual A1/A2B Receptor Blockade Improves Cardiac and Renal Outcomes in a Rat Model of Heart Failure with Preserved Ejection Fraction.

Tofovic SP, Salah EM, Smits GJ, Whalley ET, Ticho B, Deykin A, Jackson EK. Tofovic SP, et al. Among authors: whalley et. J Pharmacol Exp Ther. 2016 Feb;356(2):333-40. doi: 10.1124/jpet.115.228841. Epub 2015 Nov 19. J Pharmacol Exp Ther. 2016. PMID: 26585572 Free PMC article.

9

A new class of bradykinin antagonists: synthesis and in vitro activity of bissuccinimidoalkane peptide dimers.

Cheronis JC, Whalley ET, Nguyen KT, Eubanks SR, Allen LG, Duggan MJ, Loy SD, Bonham KA, Blodgett JK. Cheronis JC, et al. Among authors: whalley et. J Med Chem. 1992 May 1;35(9):1563-72. doi: 10.1021/jm00087a010. J Med Chem. 1992. PMID: 1578482

10

Protective effect of tonapofylline (BG9928), an adenosine A1 receptor antagonist, against cisplatin-induced acute kidney injury in rats.

Gill A, Wortham K, Costa D, Davis W, Ticho B, Whalley E. Gill A, et al. Am J Nephrol. 2009;30(6):521-6. doi: 10.1159/000248762. Epub 2009 Oct 13. Am J Nephrol. 2009. PMID: 19828940

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