Caggiano TJ - Search Results

1

Pyridobenzodiazepines: a novel class of orally active, vasopressin V2 receptor selective agonists.

Failli AA, Shumsky JS, Steffan RJ, Caggiano TJ, Williams DK, Trybulski EJ, Ning X, Lock Y, Tanikella T, Hartmann D, Chan PS, Park CH. Failli AA, et al. Among authors: caggiano tj. Bioorg Med Chem Lett. 2006 Feb 15;16(4):954-9. doi: 10.1016/j.bmcl.2005.10.107. Epub 2005 Nov 15. Bioorg Med Chem Lett. 2006. PMID: 16297621

2

The design, synthesis and physical chemical properties of novel human vasopressin V2-receptor antagonists optimized for parenteral delivery.

Ashwell MA, Bagli JF, Caggiano TJ, Chan PS, Molinari AJ, Palka C, Park CH, Rogers JF, Sherman M, Trybulski EJ, Williams DK. Ashwell MA, et al. Among authors: caggiano tj. Bioorg Med Chem Lett. 2000 Apr 17;10(8):783-6. doi: 10.1016/s0960-894x(00)00095-0. Bioorg Med Chem Lett. 2000. PMID: 10782686

3

Estrogen receptor dependent inhibitors of NF-kappaB transcriptional activation-1 synthesis and biological evaluation of substituted 2-cyanopropanoic acid derivatives: pathway selective inhibitors of NF-kappaB, a potential treatment for rheumatoid arthritis.

Caggiano TJ, Brazzale A, Ho DM, Kraml CM, Trybulski E, Chadwick CC, Chippari S, Borges-Marcucci L, Eckert A, Keith JC, Kenney T, Harnish DC. Caggiano TJ, et al. J Med Chem. 2007 Nov 1;50(22):5245-8. doi: 10.1021/jm701013k. Epub 2007 Sep 29. J Med Chem. 2007. PMID: 17902637

4

Normal-phase automated mass-directed HPLC purification of a pyrrolobenzodiazepine library with vasopressin agonist activity.

Kagan M, Chlenov M, Melnikov S, McConnell O, Bach AC 2nd, Carter G, Failli A, Caggiano TJ, Shumsky JS, Lubda D. Kagan M, et al. Among authors: caggiano tj. J Comb Chem. 2009 Jul-Aug;11(4):704-19. doi: 10.1021/cc9000407. J Comb Chem. 2009. PMID: 19459687

5

The activity of pathway-selective estrogen receptor ligands in experimental septic shock.

Opal SM, Palardy JE, Cristofaro P, Parejo N, Jhung JW, Keith JC Jr, Chippari S, Caggiano TJ, Steffan RJ, Chadwick CC, Harnish DC. Opal SM, et al. Among authors: caggiano tj. Shock. 2005 Dec;24(6):535-40. doi: 10.1097/01.shk.0000183388.90895.cb. Shock. 2005. PMID: 16317384

6

Synthesis and structure-activity relationship of a novel series of heterocyclic sulfonamide gamma-secretase inhibitors.

Pu J, Kreft AF, Aschmies SH, Atchison KP, Berkowitz J, Caggiano TJ, Chlenov M, Diamantidis G, Harrison BL, Hu Y, Huryn D, Steven Jacobsen J, Jin M, Lipinski K, Lu P, Martone RL, Morris K, Sonnenberg-Reines J, Riddell DR, Sabalski J, Sun SC, Wagner E, Wang Y, Xu Z, Zhou H, Resnick L. Pu J, et al. Among authors: caggiano tj. Bioorg Med Chem. 2009 Jul 1;17(13):4708-17. doi: 10.1016/j.bmc.2009.04.052. Epub 2009 May 3. Bioorg Med Chem. 2009. PMID: 19443228

7

Studies on new acidic azoles as glucose-lowering agents in obese, diabetic db/db mice.

Kees KL, Caggiano TJ, Steiner KE, Fitzgerald JJ Jr, Kates MJ, Christos TE, Kulishoff JM Jr, Moore RD, McCaleb ML. Kees KL, et al. Among authors: caggiano tj. J Med Chem. 1995 Feb 17;38(4):617-28. doi: 10.1021/jm00004a008. J Med Chem. 1995. PMID: 7861410

8

Structure-activity relationships of 1H-indole-7-carboxamides as a novel series of selective alpha 1-adrenoceptor agonists.

Rimele TJ, Caggiano TJ, Buckley SK, Dustman WJ, Schmid J, Heaslip RJ, Grimes D, Asselin AA. Rimele TJ, et al. Among authors: caggiano tj. Arzneimittelforschung. 1989 Feb;39(2):187-95. Arzneimittelforschung. 1989. PMID: 2567168

9

A putative sirolimus (rapamycin) effector protein.

Chen Y, Chen H, Rhoad AE, Warner L, Caggiano TJ, Failli A, Zhang H, Hsiao CL, Nakanishi K, Molnar-Kimber KL. Chen Y, et al. Among authors: caggiano tj. Biochem Biophys Res Commun. 1994 Aug 30;203(1):1-7. doi: 10.1006/bbrc.1994.2140. Biochem Biophys Res Commun. 1994. PMID: 7521160

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