Ganellin CR - Search Results

1

Partial structures of ketoconazole as modulators of the large conductance calcium-activated potassium channel (BK(Ca)).

Power EC, Ganellin CR, Benton DC. Power EC, et al. Among authors: ganellin cr. Bioorg Med Chem Lett. 2006 Feb 15;16(4):887-90. doi: 10.1016/j.bmcl.2005.11.001. Epub 2005 Dec 15. Bioorg Med Chem Lett. 2006. PMID: 16359866

2

Synthesis and structure-activity relationships of cetiedil analogues as blockers of the Ca(2+)-activated K+ permeability of erythrocytes.

Roxburgh CJ, Ganellin CR, Athmani S, Bisi A, Quaglia W, Benton DC, Shiner MA, Malik-Hall M, Haylett DG, Jenkinson DH. Roxburgh CJ, et al. Among authors: ganellin cr. J Med Chem. 2001 Sep 27;44(20):3244-53. doi: 10.1021/jm001113w. J Med Chem. 2001. PMID: 11563923

3

Enhancement of hippocampal pyramidal cell excitability by the novel selective slow-afterhyperpolarization channel blocker 3-(triphenylmethylaminomethyl)pyridine (UCL2077).

Shah MM, Javadzadeh-Tabatabaie M, Benton DC, Ganellin CR, Haylett DG. Shah MM, et al. Among authors: ganellin cr. Mol Pharmacol. 2006 Nov;70(5):1494-502. doi: 10.1124/mol.106.026625. Epub 2006 Jul 28. Mol Pharmacol. 2006. PMID: 16877678 Free PMC article.

4

Synthesis of novel ketoconazole derivatives as inhibitors of the human Pregnane X Receptor (PXR; NR1I2; also termed SXR, PAR).

Das BC, Madhukumar AV, Anguiano J, Kim S, Sinz M, Zvyaga TA, Power EC, Ganellin CR, Mani S. Das BC, et al. Among authors: ganellin cr. Bioorg Med Chem Lett. 2008 Jul 15;18(14):3974-7. doi: 10.1016/j.bmcl.2008.06.018. Epub 2008 Jun 10. Bioorg Med Chem Lett. 2008. PMID: 18583127

5

Discrimination between subtypes of apamin-sensitive Ca(2+)-activated K+ channels by gallamine and a novel bis-quaternary quinolinium cyclophane, UCL 1530.

Dunn PM, Benton DC, Campos Rosa J, Ganellin CR, Jenkinson DH. Dunn PM, et al. Among authors: ganellin cr. Br J Pharmacol. 1996 Jan;117(1):35-42. doi: 10.1111/j.1476-5381.1996.tb15151.x. Br J Pharmacol. 1996. PMID: 8825340 Free PMC article.

6

The synthesis and some pharmacological actions of the enantiomers of the K(+)-channel blocker cetiedil.

Roxburgh CJ, Ganellin CR, Shiner MA, Benton DC, Dunn PM, Ayalew Y, Jenkinson DH. Roxburgh CJ, et al. Among authors: ganellin cr. J Pharm Pharmacol. 1996 Aug;48(8):851-7. doi: 10.1111/j.2042-7158.1996.tb03986.x. J Pharm Pharmacol. 1996. PMID: 8887737

7

Differences in the actions of some blockers of the calcium-activated potassium permeability in mammalian red cells.

Benton DC, Roxburgh CJ, Ganellin CR, Shiner MA, Jenkinson DH. Benton DC, et al. Among authors: ganellin cr. Br J Pharmacol. 1999 Jan;126(1):169-78. doi: 10.1038/sj.bjp.0702292. Br J Pharmacol. 1999. PMID: 10051133 Free PMC article.

8

Synthesis and pharmacological testing of polyaminoquinolines as blockers of the apamin-sensitive Ca2+-activated K+ channel (SK(Ca)).

Fletcher DI, Ganellin CR, Piergentili A, Dunn PM, Jenkinson DH. Fletcher DI, et al. Among authors: ganellin cr. Bioorg Med Chem. 2007 Aug 15;15(16):5457-79. doi: 10.1016/j.bmc.2007.05.054. Epub 2007 May 26. Bioorg Med Chem. 2007. PMID: 17560109

9

Synthesis and quantitative structure-activity relationship of a novel series of small conductance Ca(2+)-activated K+ channel blockers related to dequalinium.

Galanakis D, Davis CA, Ganellin CR, Dunn PM. Galanakis D, et al. Among authors: ganellin cr. J Med Chem. 1996 Jan 19;39(2):359-70. doi: 10.1021/jm950520i. J Med Chem. 1996. PMID: 8558503

10

Meta-substituted aryl(thio)ethers as potent partial agonists (or antagonists) for the histamine H3 receptor lacking a nitrogen atom in the side chain.

Pelloux-Léon N, Fkyerat A, Piripitsi A, Tertiuk W, Schunack W, Stark H, Garbarg M, Ligneau X, Arrang JM, Schwartz JC, Ganellin CR. Pelloux-Léon N, et al. Among authors: ganellin cr. J Med Chem. 2004 Jun 3;47(12):3264-74. doi: 10.1021/jm031141p. J Med Chem. 2004. PMID: 15163206

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