Schirrmacher R - Search Results

1

Synthesis of 131I-labeled glucose-conjugated inhibitors of O6-methylguanine-DNA methyltransferase (MGMT) and comparison with nonconjugated inhibitors as potential tools for in vivo MGMT imaging.

Mühlhausen U, Schirrmacher R, Piel M, Lecher B, Briegert M, Piee-Staffa A, Kaina B, Rösch F. Mühlhausen U, et al. Among authors: schirrmacher r. J Med Chem. 2006 Jan 12;49(1):263-72. doi: 10.1021/jm050588q. J Med Chem. 2006. PMID: 16392811

2

An approach to the evaluation of the activity of the DNA repair enzyme O6-methylguanine-DNA-methyl-transferase in tumor tissue in vivo: syntheses of 6-benzyloxy-9-(2-[18F]fluoroethyl)-9H-purin-2-yl-amine and 6-benzyloxy-7-(2-[18F]fluoroethyl)-7H-purin-2-yl-amine.

Schirrmacher R, Nesseler E, Hamkens W, Eichhorn U, Schreckenberger M, Kaina B, Rösch F. Schirrmacher R, et al. Appl Radiat Isot. 2002 Mar;56(3):511-7. doi: 10.1016/s0969-8043(01)00155-5. Appl Radiat Isot. 2002. PMID: 11922418

3

Efficient synthesis of 2-bromo-1-[18F]fluoroethane and its application in the automated preparation of 18F-fluoroethylated compounds.

Comagic S, Piel M, Schirrmacher R, Höhnemann S, Rösch F. Comagic S, et al. Among authors: schirrmacher r. Appl Radiat Isot. 2002 Jun;56(6):847-51. doi: 10.1016/s0969-8043(01)00237-8. Appl Radiat Isot. 2002. PMID: 12102341

4

Synthesis and preliminary evaluation of (R,R)(S,S) 5-(2-(2-[4-(2-[(18)F]fluoroethoxy)phenyl]-1-methylethylamino)-1-hydroxyethyl)-benzene-1,3-diol ([(18)F]FEFE) for the in vivo visualisation and quantification of the beta2-adrenergic receptor status in lung.

Schirrmacher E, Schirrmacher R, Thews O, Dillenburg W, Helisch A, Wessler I, Buhl R, Höhnemann S, Buchholz HG, Bartenstein P, Machulla HJ, Rösch F. Schirrmacher E, et al. Among authors: schirrmacher r. Bioorg Med Chem Lett. 2003 Aug 18;13(16):2687-92. doi: 10.1016/s0960-894x(03)00538-9. Bioorg Med Chem Lett. 2003. PMID: 12873495

5

Synthesis and evaluation of fluorine-18 labeled glyburide analogs as beta-cell imaging agents.

Schmitz A, Shiue CY, Feng Q, Shiue GG, Deng S, Pourdehnad MT, Schirrmacher R, Vatamaniuk M, Doliba N, Matschinsky F, Wolf B, Rösch F, Naji A, Alavi AA. Schmitz A, et al. Among authors: schirrmacher r. Nucl Med Biol. 2004 May;31(4):483-91. doi: 10.1016/j.nucmedbio.2003.12.003. Nucl Med Biol. 2004. PMID: 15093819

6

Synthesis and evaluation of (S)-2-(2-[18F]fluoroethoxy)-4-([3-methyl-1-(2-piperidin-1-yl-phenyl)-butyl-carbamoyl]-methyl)-benzoic acid ([18F]repaglinide): a promising radioligand for quantification of pancreatic beta-cell mass with positron emission tomography (PET).

Wängler B, Schneider S, Thews O, Schirrmacher E, Comagic S, Feilen P, Schwanstecher C, Schwanstecher M, Shiue CY, Alavi A, Höhnemann S, Piel M, Rösch F, Schirrmacher R. Wängler B, et al. Among authors: schirrmacher r, schirrmacher e. Nucl Med Biol. 2004 Jul;31(5):639-47. doi: 10.1016/j.nucmedbio.2004.01.007. Nucl Med Biol. 2004. PMID: 15219283

7

Inhibition of O6-methylguanine-DNA methyltransferase by glucose-conjugated inhibitors: comparison with nonconjugated inhibitors and effect on fotemustine and temozolomide-induced cell death.

Kaina B, Mühlhausen U, Piee-Staffa A, Christmann M, Garcia Boy R, Rösch F, Schirrmacher R. Kaina B, et al. Among authors: schirrmacher r. J Pharmacol Exp Ther. 2004 Nov;311(2):585-93. doi: 10.1124/jpet.104.071316. Epub 2004 Jul 13. J Pharmacol Exp Ther. 2004. PMID: 15254145

8

Synthesis and in vitro evaluation of (S)-2-([11C]methoxy)-4-[3-methyl-1-(2-piperidine-1-yl-phenyl)-butyl-carbamoyl]-benzoic acid ([11C]methoxy-repaglinide): a potential beta-cell imaging agent.

Wängler B, Beck C, Shiue CY, Schneider S, Schwanstecher C, Schwanstecher M, Feilen PJ, Alavi A, Rösch F, Schirrmacher R. Wängler B, et al. Among authors: schirrmacher r. Bioorg Med Chem Lett. 2004 Oct 18;14(20):5205-9. doi: 10.1016/j.bmcl.2004.07.059. Bioorg Med Chem Lett. 2004. PMID: 15380228

9

Parametric mapping of binding in human brain of D2 receptor ligands of different affinities.

Siessmeier T, Zhou Y, Buchholz HG, Landvogt C, Vernaleken I, Piel M, Schirrmacher R, Rösch F, Schreckenberger M, Wong DF, Cumming P, Gründer G, Bartenstein P. Siessmeier T, et al. Among authors: schirrmacher r. J Nucl Med. 2005 Jun;46(6):964-72. J Nucl Med. 2005. PMID: 15937307 Free article.

10

In vitro and in vivo evaluation of novel glibenclamide derivatives as imaging agents for the non-invasive assessment of the pancreatic islet cell mass in animals and humans.

Schneider S, Feilen PJ, Schreckenberger M, Schwanstecher M, Schwanstecher C, Buchholz HG, Thews O, Oberholzer K, Korobeynikov A, Bauman A, Comagic S, Piel M, Schirrmacher E, Shiue CY, Alavi AA, Bartenstein P, Rösch F, Weber MM, Klein HH, Schirrmacher R. Schneider S, et al. Among authors: schirrmacher r, schirrmacher e. Exp Clin Endocrinol Diabetes. 2005 Jul;113(7):388-95. doi: 10.1055/s-2005-865711. Exp Clin Endocrinol Diabetes. 2005. PMID: 16025400

Save citations to file

Email citations

Send citations to clipboard

Add to Collections

Add to My Bibliography

Create a file for external citation management software

Your saved search

Your RSS Feed

My Custom Filters

Publication date

Text availability

Article attribute

Article type

Article Language

Species

Sex

Age

Other

149 results

Search Page

Filters