Marcopulos N - Search Results

1

Synthesis and selective class III antiarrhythmic activity of novel N-heteroaralkyl-substituted 1-(aryloxy)-2-propanolamine and related propylamine derivatives.

Butera JA, Spinelli W, Anantharaman V, Marcopulos N, Parsons RW, Moubarak IF, Cullinan C, Bagli JF. Butera JA, et al. Among authors: marcopulos n. J Med Chem. 1991 Nov;34(11):3212-28. doi: 10.1021/jm00115a010. J Med Chem. 1991. PMID: 1956040

2

Design and synthesis of potent, selective inhibitors of endothelin-converting enzyme.

Wallace EM, Moliterni JA, Moskal MA, Neubert AD, Marcopulos N, Stamford LB, Trapani AJ, Savage P, Chou M, Jeng AY. Wallace EM, et al. Among authors: marcopulos n. J Med Chem. 1998 Apr 23;41(9):1513-23. doi: 10.1021/jm970787c. J Med Chem. 1998. PMID: 9554884

3

Perhydroquinolylbenzamides as novel inhibitors of 11beta-hydroxysteroid dehydrogenase type 1.

Coppola GM, Kukkola PJ, Stanton JL, Neubert AD, Marcopulos N, Bilci NA, Wang H, Tomaselli HC, Tan J, Aicher TD, Knorr DC, Jeng AY, Dardik B, Chatelain RE. Coppola GM, et al. Among authors: marcopulos n. J Med Chem. 2005 Oct 20;48(21):6696-712. doi: 10.1021/jm058228q. J Med Chem. 2005. PMID: 16220986

4

Discovery of orally active carboxylic acid derivatives of 2-phenyl-5-trifluoromethyloxazole-4-carboxamide as potent diacylglycerol acyltransferase-1 inhibitors for the potential treatment of obesity and diabetes.

Qian Y, Wertheimer SJ, Ahmad M, Cheung AW, Firooznia F, Hamilton MM, Hayden S, Li S, Marcopulos N, McDermott L, Tan J, Yun W, Guo L, Pamidimukkala A, Chen Y, Huang KS, Ramsey GB, Whittard T, Conde-Knape K, Taub R, Rondinone CM, Tilley J, Bolin D. Qian Y, et al. Among authors: marcopulos n. J Med Chem. 2011 Apr 14;54(7):2433-46. doi: 10.1021/jm101580m. Epub 2011 Mar 17. J Med Chem. 2011. PMID: 21413799

5

7-Phenyl-pyrido[2,3-d]pyrimidine-2,4-diamines: novel and highly selective protein tyrosine phosphatase 1B inhibitors.

Cheung AW, Banner B, Bose J, Kim K, Li S, Marcopulos N, Orzechowski L, Sergi JA, Thakkar KC, Wang BB, Yun W, Zwingelstein C, Berthel S, Olivier AR. Cheung AW, et al. Among authors: marcopulos n. Bioorg Med Chem Lett. 2012 Dec 15;22(24):7518-22. doi: 10.1016/j.bmcl.2012.10.035. Epub 2012 Oct 16. Bioorg Med Chem Lett. 2012. PMID: 23122867

6

Discovery of benzothiazole-based adenosine A2B receptor antagonists with improved A2A selectivity.

Firooznia F, Cheung AW, Brinkman J, Grimsby J, Gubler ML, Hamid R, Marcopulos N, Ramsey G, Tan J, Wen Y, Sarabu R. Firooznia F, et al. Among authors: marcopulos n. Bioorg Med Chem Lett. 2011 Apr 1;21(7):1933-6. doi: 10.1016/j.bmcl.2011.02.053. Epub 2011 Feb 17. Bioorg Med Chem Lett. 2011. PMID: 21388809

7

4-Substituted-7-N-alkyl-N-acetyl 2-aminobenzothiazole amides: drug-like and non-xanthine based A2B adenosine receptor antagonists.

Cheung AW, Brinkman J, Firooznia F, Flohr A, Grimsby J, Gubler ML, Guertin K, Hamid R, Marcopulos N, Norcross RD, Qi L, Ramsey G, Tan J, Wen Y, Sarabu R. Cheung AW, et al. Among authors: marcopulos n. Bioorg Med Chem Lett. 2010 Jul 15;20(14):4140-6. doi: 10.1016/j.bmcl.2010.05.056. Epub 2010 May 20. Bioorg Med Chem Lett. 2010. PMID: 20541935

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