Okun IM - Search Results

1

Synthesis of cycloalkane-annelated 3-phenylsulfonyl-pyrazolo[1,5-a]pyrimidines and their evaluation as 5-HT6 receptor antagonists.

Ivachtchenko AV, Dmitriev DE, Golovina ES, Dubrovskaya ES, Kadieva MG, Koryakova AG, Kysil VM, Mitkin OD, Tkachenko SE, Okun IM, Vorobiov AA. Ivachtchenko AV, et al. Among authors: okun im. Bioorg Med Chem Lett. 2010 Apr 1;20(7):2133-6. doi: 10.1016/j.bmcl.2010.02.046. Epub 2010 Feb 14. Bioorg Med Chem Lett. 2010. PMID: 20207539

2

1,3-Dioxo-4-methyl-2,3-dihydro-1H-pyrrolo[3,4-c]quinolines as potent caspase-3 inhibitors.

Kravchenko DV, Kysil VV, Ilyn AP, Tkachenko SE, Maliarchouk S, Okun IM, Ivachtchenko AV. Kravchenko DV, et al. Among authors: okun im. Bioorg Med Chem Lett. 2005 Apr 1;15(7):1841-5. doi: 10.1016/j.bmcl.2005.02.027. Bioorg Med Chem Lett. 2005. PMID: 15780618

3

Synthesis and structure-activity relationship of 4-substituted 2-(2-acetyloxyethyl)-8-(morpholine-4-sulfonyl)pyrrolo[3,4-c]quinoline-1,3-diones as potent caspase-3 inhibitors.

Kravchenko DV, Kuzovkova YA, Kysil VM, Tkachenko SE, Maliarchouk S, Okun IM, Balakin KV, Ivachtchenko AV. Kravchenko DV, et al. Among authors: okun im. J Med Chem. 2005 Jun 2;48(11):3680-3. doi: 10.1021/jm048987t. J Med Chem. 2005. PMID: 15916416

4

Pyrrolo[3,4-c]quinoline-1,3-diones as potent caspase-3 inhibitors. Synthesis and SAR of 2-substituted 4-methyl-8-(morpholine-4-sulfonyl)-pyrrolo[3,4-c]quinoline-1,3-diones.

Kravchenko DV, Kysil VM, Tkachenko SE, Maliarchouk S, Okun IM, Ivachtchenko AV. Kravchenko DV, et al. Among authors: okun im. Eur J Med Chem. 2005 Dec;40(12):1377-83. doi: 10.1016/j.ejmech.2005.07.011. Epub 2005 Sep 15. Eur J Med Chem. 2005. PMID: 16169127

5

Synthesis and biological evaluation of novel gamma-carboline analogues of Dimebon as potent 5-HT6 receptor antagonists.

Ivachtchenko AV, Frolov EB, Mitkin OD, Kysil VM, Khvat AV, Okun IM, Tkachenko SE. Ivachtchenko AV, et al. Among authors: okun im. Bioorg Med Chem Lett. 2009 Jun 15;19(12):3183-7. doi: 10.1016/j.bmcl.2009.04.128. Epub 2009 May 3. Bioorg Med Chem Lett. 2009. PMID: 19443217

6

8-Sulfonyl-substituted tetrahydro-1H-pyrido[4,3-b]indoles as 5-HT6 receptor antagonists.

Ivachtchenko AV, Mitkin OD, Tkachenko SE, Okun IM, Kysil VM. Ivachtchenko AV, et al. Among authors: okun im. Eur J Med Chem. 2010 Feb;45(2):782-9. doi: 10.1016/j.ejmech.2009.10.035. Epub 2009 Oct 31. Eur J Med Chem. 2010. PMID: 19939513

7

Synthesis and biological activity of 5-styryl and 5-phenethyl-substituted 2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indoles.

Ivachtchenko AV, Frolov EB, Mitkin OD, Tkachenko SE, Okun IM, Khvat AV. Ivachtchenko AV, et al. Among authors: okun im. Bioorg Med Chem Lett. 2010 Jan 1;20(1):78-82. doi: 10.1016/j.bmcl.2009.11.037. Epub 2009 Nov 14. Bioorg Med Chem Lett. 2010. PMID: 19945877

8

Solution phase parallel synthesis of substituted 3-phenylsulfonyl-[1,2,3]triazolo[1,5-a]quinazolines: selective serotonin 5-HT(6) receptor antagonists.

Ivachtchenko AV, Golovina ES, Kadieva MG, Koryakova AG, Kovalenko SM, Mitkin OD, Okun IM, Ravnyeyko IM, Tkachenko SE, Zaremba OV. Ivachtchenko AV, et al. Among authors: okun im. J Comb Chem. 2010 Jul 12;12(4):445-52. doi: 10.1021/cc1000049. J Comb Chem. 2010. PMID: 20349953

9

Synthesis and biological study of 3-(phenylsulfonyl)thieno[2,3-e][1,2,3]triazolo[1,5-a]pyrimidines as potent and selective serotonin 5-HT6 receptor antagonists.

Ivachtchenko AV, Golovina ES, Kadieva MG, Koryakova AG, Kovalenko SM, Mitkin OD, Okun IM, Ravnyeyko IM, Tkachenko SE, Zaremba OV. Ivachtchenko AV, et al. Among authors: okun im. Bioorg Med Chem. 2010 Jul 15;18(14):5282-90. doi: 10.1016/j.bmc.2010.05.051. Epub 2010 May 24. Bioorg Med Chem. 2010. PMID: 20541425

10

(3-Phenylsulfonylcycloalkano[e and d]pyrazolo[1,5-a]pyrimidin-2-yl)amines: potent and selective antagonists of the serotonin 5-HT6 receptor.

Ivachtchenko AV, Dmitriev DE, Golovina ES, Kadieva MG, Koryakova AG, Kysil VM, Mitkin OD, Okun IM, Tkachenko SE, Vorobiev AA. Ivachtchenko AV, et al. Among authors: okun im. J Med Chem. 2010 Jul 22;53(14):5186-96. doi: 10.1021/jm100350r. J Med Chem. 2010. PMID: 20560595

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