Design and synthesis of an orally bioavailable and selective peptide epoxyketone proteasome inhibitor (PR-047).
Zhou HJ, Aujay MA, Bennett MK, Dajee M, Demo SD, Fang Y, Ho MN, Jiang J, Kirk CJ, Laidig GJ, Lewis ER, Lu Y, Muchamuel T, Parlati F, Ring E, Shenk KD, Shields J, Shwonek PJ, Stanton T, Sun CM, Sylvain C, Woo TM, Yang J.
Zhou HJ, et al. Among authors: kirk cj.
J Med Chem. 2009 May 14;52(9):3028-38. doi: 10.1021/jm801329v.
J Med Chem. 2009.
PMID: 19348473