Overkleeft HS - Search Results

1

Discovery of a potent and highly β1 specific proteasome inhibitor from a focused library of urea-containing peptide vinyl sulfones and peptide epoxyketones.

van der Linden WA, Willems LI, Shabaneh TB, Li N, Ruben M, Florea BI, van der Marel GA, Kaiser M, Kisselev AF, Overkleeft HS. van der Linden WA, et al. Among authors: overkleeft hs. Org Biomol Chem. 2012 Jan 7;10(1):181-94. doi: 10.1039/c1ob06554h. Epub 2011 Nov 22. Org Biomol Chem. 2012. PMID: 22105930 Free PMC article.

2

Extended peptide-based inhibitors efficiently target the proteasome and reveal overlapping specificities of the catalytic beta-subunits.

Kessler BM, Tortorella D, Altun M, Kisselev AF, Fiebiger E, Hekking BG, Ploegh HL, Overkleeft HS. Kessler BM, et al. Among authors: overkleeft hs. Chem Biol. 2001 Sep;8(9):913-29. doi: 10.1016/s1074-5521(01)00069-2. Chem Biol. 2001. PMID: 11564559

3

Extending solid-phase methods in inorganic synthesis: the first dinuclear platinum complex synthesised via the solid phase.

van Zutphen S, Robillard MS, van der Marel GA, Overkleeft HS, den Dulk H, Brouwer J, Reedijk J. van Zutphen S, et al. Among authors: overkleeft hs. Chem Commun (Camb). 2003 Mar 7;(5):634-5. doi: 10.1039/b212388f. Chem Commun (Camb). 2003. PMID: 12669861

4

Ph2SO/Tf2O: a powerful promotor system in chemoselective glycosylations using thioglycosides.

Codée JD, Litjens RE, den Heeten R, Overkleeft HS, van Boom JH, van der Marel GA. Codée JD, et al. Among authors: overkleeft hs. Org Lett. 2003 May 1;5(9):1519-22. doi: 10.1021/ol034312t. Org Lett. 2003. PMID: 12713313

5

Sequential one-pot glycosylations using 1-hydroxyl and 1-thiodonors.

Codée JD, van den Bos LJ, Litjens RE, Overkleeft HS, van Boom JH, van der Marel GA. Codée JD, et al. Among authors: overkleeft hs. Org Lett. 2003 May 29;5(11):1947-50. doi: 10.1021/ol034528v. Org Lett. 2003. PMID: 12762693

6

The caspase-like sites of proteasomes, their substrate specificity, new inhibitors and substrates, and allosteric interactions with the trypsin-like sites.

Kisselev AF, Garcia-Calvo M, Overkleeft HS, Peterson E, Pennington MW, Ploegh HL, Thornberry NA, Goldberg AL. Kisselev AF, et al. Among authors: overkleeft hs. J Biol Chem. 2003 Sep 19;278(38):35869-77. doi: 10.1074/jbc.M303725200. Epub 2003 Jun 18. J Biol Chem. 2003. PMID: 12815064 Free article.

7

The use of a mannitol-derived fused oxacycle as a combinatorial scaffold.

Timmer MS, Verdoes M, Sliedregt LA, van der Marel GA, van Boom JH, Overkleeft HS. Timmer MS, et al. Among authors: overkleeft hs. J Org Chem. 2003 Nov 28;68(24):9406-11. doi: 10.1021/jo0349429. J Org Chem. 2003. PMID: 14629165

8

A novel strategy towards the synthesis of orthogonally functionalised 4-aminoglycosides.

van den Bos LJ, Codée JD, van Boom JH, Overkleeft HS, van der Marel GA. van den Bos LJ, et al. Among authors: overkleeft hs. Org Biomol Chem. 2003 Dec 7;1(23):4160-5. doi: 10.1039/b309823k. Epub 2003 Oct 21. Org Biomol Chem. 2003. PMID: 14685319

9

Design, synthesis, and evaluation of sugar amino acid based inhibitors of protein prenyl transferases PFT and PGGT-1.

El Oualid F, Burm BE, Leroy IM, Cohen LH, van Boom JH, van den Elst H, Overkleeft HS, van der Marel GA, Overhand M. El Oualid F, et al. Among authors: overkleeft hs. J Med Chem. 2004 Jul 29;47(16):3920-3. doi: 10.1021/jm049927q. J Med Chem. 2004. PMID: 15267228

10

Alkylated sugar amino acids: a new entry toward highly functionalized dipeptide isosters.

Raunkjaer M, El Oualid F, van der Marel GA, Overkleeft HS, Overhand M. Raunkjaer M, et al. Among authors: overkleeft hs. Org Lett. 2004 Sep 2;6(18):3167-70. doi: 10.1021/ol048750r. Org Lett. 2004. PMID: 15330614

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