Gilon C - Search Results

1

Intestinal permeability of cyclic peptides: common key backbone motifs identified.

Beck JG, Chatterjee J, Laufer B, Kiran MU, Frank AO, Neubauer S, Ovadia O, Greenberg S, Gilon C, Hoffman A, Kessler H. Beck JG, et al. Among authors: gilon c. J Am Chem Soc. 2012 Jul 25;134(29):12125-33. doi: 10.1021/ja303200d. Epub 2012 Jul 12. J Am Chem Soc. 2012. PMID: 22737969

2

Comparison of the conformation of active and nonactive backbone cyclic analogs of substance P as a tool to elucidate features of the bioactive conformation: NMR and molecular dynamics in DMSO and water.

Grdadolnik SG, Mierke DF, Byk G, Zeltser I, Gilon C, Kessler H. Grdadolnik SG, et al. Among authors: gilon c. J Med Chem. 1994 Jul 8;37(14):2145-52. doi: 10.1021/jm00040a005. J Med Chem. 1994. PMID: 7518522

3

Structure-activity relationship of the ring portion in backbone-cyclic C-terminal hexapeptide analogs of substance P. NMR and molecular dynamics.

Behrens S, Mathä B, Bitan G, Gilon C, Kessler H. Behrens S, et al. Among authors: gilon c. Int J Pept Protein Res. 1996 Dec;48(6):569-79. doi: 10.1111/j.1399-3011.1996.tb00876.x. Int J Pept Protein Res. 1996. PMID: 8985790

4

Multiple N-methylation by a designed approach enhances receptor selectivity.

Chatterjee J, Ovadia O, Zahn G, Marinelli L, Hoffman A, Gilon C, Kessler H. Chatterjee J, et al. Among authors: gilon c. J Med Chem. 2007 Nov 29;50(24):5878-81. doi: 10.1021/jm701044r. Epub 2007 Nov 1. J Med Chem. 2007. PMID: 17973471

5

Effect of structural and conformation modifications, including backbone cyclization, of hydrophilic hexapeptides on their intestinal permeability and enzymatic stability.

Hess S, Ovadia O, Shalev DE, Senderovich H, Qadri B, Yehezkel T, Salitra Y, Sheynis T, Jelinek R, Gilon C, Hoffman A. Hess S, et al. Among authors: gilon c. J Med Chem. 2007 Nov 29;50(24):6201-11. doi: 10.1021/jm070836d. Epub 2007 Nov 6. J Med Chem. 2007. PMID: 17983214

6

Backbone cyclic peptidomimetic melanocortin-4 receptor agonist as a novel orally administrated drug lead for treating obesity.

Hess S, Linde Y, Ovadia O, Safrai E, Shalev DE, Swed A, Halbfinger E, Lapidot T, Winkler I, Gabinet Y, Faier A, Yarden D, Xiang Z, Portillo FP, Haskell-Luevano C, Gilon C, Hoffman A. Hess S, et al. Among authors: gilon c. J Med Chem. 2008 Feb 28;51(4):1026-34. doi: 10.1021/jm701093y. Epub 2008 Jan 26. J Med Chem. 2008. PMID: 18220330

7

Improving oral bioavailability of peptides by multiple N-methylation: somatostatin analogues.

Biron E, Chatterjee J, Ovadia O, Langenegger D, Brueggen J, Hoyer D, Schmid HA, Jelinek R, Gilon C, Hoffman A, Kessler H. Biron E, et al. Among authors: gilon c. Angew Chem Int Ed Engl. 2008;47(14):2595-9. doi: 10.1002/anie.200705797. Angew Chem Int Ed Engl. 2008. PMID: 18297660 No abstract available.

8

N-methylation of peptides: a new perspective in medicinal chemistry.

Chatterjee J, Gilon C, Hoffman A, Kessler H. Chatterjee J, et al. Among authors: gilon c. Acc Chem Res. 2008 Oct;41(10):1331-42. doi: 10.1021/ar8000603. Epub 2008 Jul 18. Acc Chem Res. 2008. PMID: 18636716

9

Structure-activity relationship and metabolic stability studies of backbone cyclization and N-methylation of melanocortin peptides.

Linde Y, Ovadia O, Safrai E, Xiang Z, Portillo FP, Shalev DE, Haskell-Luevano C, Hoffman A, Gilon C. Linde Y, et al. Among authors: gilon c. Biopolymers. 2008;90(5):671-82. doi: 10.1002/bip.21057. Biopolymers. 2008. PMID: 18655141 Free PMC article.

10

N-methylated cyclic pentapeptides as template structures.

Chatterjee J, Ovadia O, Gilon C, Hoffman A, Mierke D, Kessler H. Chatterjee J, et al. Among authors: gilon c. Adv Exp Med Biol. 2009;611:109-10. doi: 10.1007/978-0-387-73657-0_48. Adv Exp Med Biol. 2009. PMID: 19400115 No abstract available.

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