Schaible AM - Search Results

1

Modified acidic nonsteroidal anti-inflammatory drugs as dual inhibitors of mPGES-1 and 5-LOX.

Elkady M, Nieß R, Schaible AM, Bauer J, Luderer S, Ambrosi G, Werz O, Laufer SA. Elkady M, et al. Among authors: schaible am. J Med Chem. 2012 Oct 25;55(20):8958-62. doi: 10.1021/jm3010543. Epub 2012 Oct 9. J Med Chem. 2012. PMID: 22992107

2

Identification of new γ-hydroxybutenolides that preferentially inhibit the activity of mPGES-1.

De Simone R, Bruno I, Riccio R, Stadler K, Bauer J, Schaible AM, Laufer S, Werz O. De Simone R, et al. Among authors: schaible am. Bioorg Med Chem. 2012 Aug 15;20(16):5012-6. doi: 10.1016/j.bmc.2012.06.032. Epub 2012 Jun 23. Bioorg Med Chem. 2012. PMID: 22795900

3

Potent inhibition of human 5-lipoxygenase and microsomal prostaglandin E₂ synthase-1 by the anti-carcinogenic and anti-inflammatory agent embelin.

Schaible AM, Traber H, Temml V, Noha SM, Filosa R, Peduto A, Weinigel C, Barz D, Schuster D, Werz O. Schaible AM, et al. Biochem Pharmacol. 2013 Aug 15;86(4):476-86. doi: 10.1016/j.bcp.2013.04.015. Epub 2013 Apr 24. Biochem Pharmacol. 2013. PMID: 23623753

4

Discovery and biological evaluation of novel 1,4-benzoquinone and related resorcinol derivatives that inhibit 5-lipoxygenase.

Filosa R, Peduto A, Aparoy P, Schaible AM, Luderer S, Krauth V, Petronzi C, Massa A, de Rosa M, Reddanna P, Werz O. Filosa R, et al. Among authors: schaible am. Eur J Med Chem. 2013 Sep;67:269-79. doi: 10.1016/j.ejmech.2013.06.039. Epub 2013 Jun 27. Eur J Med Chem. 2013. PMID: 23871907

5

Indirubin core structure of glycogen synthase kinase-3 inhibitors as novel chemotype for intervention with 5-lipoxygenase.

Pergola C, Gaboriaud-Kolar N, Jestädt N, König S, Kritsanida M, Schaible AM, Li H, Garscha U, Weinigel C, Barz D, Albring KF, Huber O, Skaltsounis AL, Werz O. Pergola C, et al. Among authors: schaible am. J Med Chem. 2014 May 8;57(9):3715-23. doi: 10.1021/jm401740w. Epub 2014 Apr 17. J Med Chem. 2014. PMID: 24697244

6

Novel series of benzoquinones with high potency against 5-lipoxygenase in human polymorphonuclear leukocytes.

Filosa R, Peduto A, Schaible AM, Krauth V, Weinigel C, Barz D, Petronzi C, Bruno F, Roviezzo F, Spaziano G, D'Agostino B, De Rosa M, Werz O. Filosa R, et al. Among authors: schaible am. Eur J Med Chem. 2015 Apr 13;94:132-9. doi: 10.1016/j.ejmech.2015.02.042. Epub 2015 Feb 24. Eur J Med Chem. 2015. PMID: 25765759

7

Elucidation of the molecular mechanism and the efficacy in vivo of a novel 1,4-benzoquinone that inhibits 5-lipoxygenase.

Schaible AM, Filosa R, Temml V, Krauth V, Matteis M, Peduto A, Bruno F, Luderer S, Roviezzo F, Di Mola A, de Rosa M, D'Agostino B, Weinigel C, Barz D, Koeberle A, Pergola C, Schuster D, Werz O. Schaible AM, et al. Br J Pharmacol. 2014 May;171(9):2399-412. doi: 10.1111/bph.12592. Br J Pharmacol. 2014. PMID: 24467325 Free PMC article.

8

Pharmacophore-based discovery of a novel cytosolic phospholipase A(2)α inhibitor.

Noha SM, Jazzar B, Kuehnl S, Rollinger JM, Stuppner H, Schaible AM, Werz O, Wolber G, Schuster D. Noha SM, et al. Among authors: schaible am. Bioorg Med Chem Lett. 2012 Jan 15;22(2):1202-7. doi: 10.1016/j.bmcl.2011.11.093. Epub 2011 Nov 30. Bioorg Med Chem Lett. 2012. PMID: 22192589 Free PMC article.

9

Caulerpenyne and related bis-enol esters are novel-type inhibitors of human 5-lipoxygenase.

Richter P, Schubert G, Schaible AM, Cavas L, Werz O, Pohnert G. Richter P, et al. Among authors: schaible am. ChemMedChem. 2014 Aug;9(8):1655-9. doi: 10.1002/cmdc.201402065. Epub 2014 Apr 11. ChemMedChem. 2014. PMID: 24729578

10

A novel C(28)-hydroxylated lupeolic acid suppresses the biosynthesis of eicosanoids through inhibition of cytosolic phospholipase A(2).

Verhoff M, Seitz S, Northoff H, Jauch J, Schaible AM, Werz O. Verhoff M, et al. Among authors: schaible am. Biochem Pharmacol. 2012 Sep 1;84(5):681-91. doi: 10.1016/j.bcp.2012.06.016. Epub 2012 Jun 23. Biochem Pharmacol. 2012. PMID: 22732453

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