Izumi M - Search Results

1

Arylpiperazines as fatty acid transport protein 1 (FATP1) inhibitors with improved potency and pharmacokinetic properties.

Matsufuji T, Ikeda M, Naito A, Hirouchi M, Kanda S, Izumi M, Harada J, Shinozuka T. Matsufuji T, et al. Among authors: izumi m. Bioorg Med Chem Lett. 2013 May 1;23(9):2560-5. doi: 10.1016/j.bmcl.2013.02.116. Epub 2013 Mar 7. Bioorg Med Chem Lett. 2013. PMID: 23528296

2

Discovery and optimization of novel fatty acid transport protein 1 (FATP1) inhibitors.

Matsufuji T, Ikeda M, Naito A, Hirouchi M, Takakusa H, Kanda S, Izumi M, Harada J, Shinozuka T. Matsufuji T, et al. Among authors: izumi m. Bioorg Med Chem Lett. 2012 Aug 1;22(15):5067-70. doi: 10.1016/j.bmcl.2012.05.130. Epub 2012 Jun 19. Bioorg Med Chem Lett. 2012. PMID: 22749869

3

Discovery of novel chiral diazepines as bombesin receptor subtype-3 (BRS-3) agonists with low brain penetration.

Matsufuji T, Shimada K, Kobayashi S, Kawamura A, Fujimoto T, Arita T, Hara T, Konishi M, Abe-Ohya R, Izumi M, Sogawa Y, Nagai Y, Yoshida K, Takahashi H. Matsufuji T, et al. Among authors: izumi m. Bioorg Med Chem Lett. 2014 Feb 1;24(3):750-5. doi: 10.1016/j.bmcl.2013.12.106. Epub 2014 Jan 2. Bioorg Med Chem Lett. 2014. PMID: 24412111

4

Synthesis and biological evaluation of novel chiral diazepine derivatives as bombesin receptor subtype-3 (BRS-3) agonists incorporating an antedrug approach.

Matsufuji T, Shimada K, Kobayashi S, Ichikawa M, Kawamura A, Fujimoto T, Arita T, Hara T, Konishi M, Abe-Ohya R, Izumi M, Sogawa Y, Nagai Y, Yoshida K, Abe Y, Kimura T, Takahashi H. Matsufuji T, et al. Among authors: izumi m. Bioorg Med Chem. 2015 Jan 1;23(1):89-104. doi: 10.1016/j.bmc.2014.11.018. Epub 2014 Nov 21. Bioorg Med Chem. 2015. PMID: 25497965

5

Discovery of a Novel Class of ERRα Agonists.

Shinozuka T, Ito S, Kimura T, Izumi M, Wakabayashi K. Shinozuka T, et al. Among authors: izumi m. ACS Med Chem Lett. 2021 Apr 21;12(5):817-821. doi: 10.1021/acsmedchemlett.1c00100. eCollection 2021 May 13. ACS Med Chem Lett. 2021. PMID: 34055231 Free PMC article.

6

Discovery of novel PTHR1 antagonists: Design, synthesis, and structure activity relationships.

Arai Y, Kiyotsuka Y, Shimada K, Oyama K, Izumi M. Arai Y, et al. Among authors: izumi m. Bioorg Med Chem Lett. 2019 Sep 15;29(18):2613-2616. doi: 10.1016/j.bmcl.2019.07.052. Epub 2019 Jul 29. Bioorg Med Chem Lett. 2019. PMID: 31383587

7

Identification of molecular target of AMP-activated protein kinase activator by affinity purification and mass spectrometry.

Kosaka T, Okuyama R, Sun W, Ogata T, Harada J, Araki K, Izumi M, Yoshida T, Okuno A, Fujiwara T, Ohsumi J, Ichikawa K. Kosaka T, et al. Among authors: izumi m. Anal Chem. 2005 Apr 1;77(7):2050-5. doi: 10.1021/ac0484631. Anal Chem. 2005. PMID: 15801737

8

Lead optimization of pyrido[2,3-d][1]benzazepin-6-one derivatives leading to the discovery of a potent, selective, and orally available human parathyroid hormone receptor 1 (hPTHR1) antagonist (DS69910557).

Arai Y, Kiyotsuka Y, Nagamochi M, Oyama K, Izumi M. Arai Y, et al. Among authors: izumi m. Bioorg Med Chem. 2022 Jun 15;64:116763. doi: 10.1016/j.bmc.2022.116763. Epub 2022 Apr 22. Bioorg Med Chem. 2022. PMID: 35487102

9

Synthesis and biological evaluation of novel imidazol-1-ylacetic acid derivatives as non-brain penetrant bombesin receptor subtype-3 (BRS-3) agonists.

Kiyotsuka Y, Shimada K, Kobayashi S, Suzuki M, Akiu M, Asano M, Sogawa Y, Hara T, Konishi M, Abe-Ohya R, Izumi M, Nagai Y, Yoshida K, Abe Y, Takamori H, Takahashi H. Kiyotsuka Y, et al. Among authors: izumi m. Bioorg Med Chem Lett. 2016 Sep 1;26(17):4205-10. doi: 10.1016/j.bmcl.2016.07.056. Epub 2016 Jul 25. Bioorg Med Chem Lett. 2016. PMID: 27491709

10

Discovery of novel, potent, and orally bioavailable pyrido[2,3-d][1]benzazepin-6-one antagonists for parathyroid hormone receptor 1.

Arai Y, Kiyotsuka Y, Kagechika K, Nishi T, Inui M, Nagamochi M, Oyama K, Izumi M. Arai Y, et al. Among authors: izumi m. Bioorg Med Chem. 2020 Jun 1;28(11):115524. doi: 10.1016/j.bmc.2020.115524. Epub 2020 Apr 22. Bioorg Med Chem. 2020. PMID: 32345459

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