Granchi C - Search Results

1

Estrogen receptors alpha (ERα) and beta (ERβ): subtype-selective ligands and clinical potential.

Paterni I, Granchi C, Katzenellenbogen JA, Minutolo F. Paterni I, et al. Among authors: granchi c. Steroids. 2014 Nov;90:13-29. doi: 10.1016/j.steroids.2014.06.012. Epub 2014 Jun 24. Steroids. 2014. PMID: 24971815 Free PMC article. Review.

2

Identification of New GSK3β Inhibitors through a Consensus Machine Learning-Based Virtual Screening.

Galati S, Di Stefano M, Bertini S, Granchi C, Giordano A, Gado F, Macchia M, Tuccinardi T, Poli G. Galati S, et al. Among authors: granchi c. Int J Mol Sci. 2023 Dec 7;24(24):17233. doi: 10.3390/ijms242417233. Int J Mol Sci. 2023. PMID: 38139062 Free PMC article.

3

alpha-Naphthylaminopropan-2-ol Derivatives as BACE1 Inhibitors.

Asso V, Ghilardi E, Bertini S, Digiacomo M, Granchi C, Minutolo F, Rapposelli S, Bortolato A, Moro S, Macchia M. Asso V, et al. Among authors: granchi c. ChemMedChem. 2008 Oct;3(10):1530-4. doi: 10.1002/cmdc.200800162. ChemMedChem. 2008. PMID: 18781572 No abstract available.

4

Structural evolutions of salicylaldoximes as selective agonists for estrogen receptor beta.

Minutolo F, Bertini S, Granchi C, Marchitiello T, Prota G, Rapposelli S, Tuccinardi T, Martinelli A, Gunther JR, Carlson KE, Katzenellenbogen JA, Macchia M. Minutolo F, et al. Among authors: granchi c. J Med Chem. 2009 Feb 12;52(3):858-67. doi: 10.1021/jm801458t. J Med Chem. 2009. PMID: 19128016

5

Bioreductively activated lysyl oxidase inhibitors against hypoxic tumours.

Granchi C, Funaioli T, Erler JT, Giaccia AJ, Macchia M, Minutolo F. Granchi C, et al. ChemMedChem. 2009 Oct;4(10):1590-4. doi: 10.1002/cmdc.200900247. ChemMedChem. 2009. PMID: 19685543 Free PMC article. No abstract available.

6

Inhibitors of lactate dehydrogenase isoforms and their therapeutic potentials.

Granchi C, Bertini S, Macchia M, Minutolo F. Granchi C, et al. Curr Med Chem. 2010;17(7):672-97. doi: 10.2174/092986710790416263. Curr Med Chem. 2010. PMID: 20088761 Review.

7

BACE1 inhibitory activities of enantiomerically pure, variously substituted N-(3-(4-benzhydrylpiperazin-1-yl)-2-hydroxypropyl) arylsulfonamides.

Bertini S, Ghilardi E, Asso V, Granchi C, Minutolo F, Pineschi M, Di Bussolo V, Bortolato A, Moro S, Saba A, Macchia M. Bertini S, et al. Among authors: granchi c. Bioorg Med Chem. 2010 Nov 15;18(22):7991-6. doi: 10.1016/j.bmc.2010.09.032. Epub 2010 Sep 18. Bioorg Med Chem. 2010. PMID: 20934348

8

Discovery of N-hydroxyindole-based inhibitors of human lactate dehydrogenase isoform A (LDH-A) as starvation agents against cancer cells.

Granchi C, Roy S, Giacomelli C, Macchia M, Tuccinardi T, Martinelli A, Lanza M, Betti L, Giannaccini G, Lucacchini A, Funel N, León LG, Giovannetti E, Peters GJ, Palchaudhuri R, Calvaresi EC, Hergenrother PJ, Minutolo F. Granchi C, et al. J Med Chem. 2011 Mar 24;54(6):1599-612. doi: 10.1021/jm101007q. Epub 2011 Feb 18. J Med Chem. 2011. PMID: 21332213

9

Selective and potent agonists for estrogen receptor beta derived from molecular refinements of salicylaldoximes.

Bertini S, De Cupertinis A, Granchi C, Bargagli B, Tuccinardi T, Martinelli A, Macchia M, Gunther JR, Carlson KE, Katzenellenbogen JA, Minutolo F. Bertini S, et al. Among authors: granchi c. Eur J Med Chem. 2011 Jun;46(6):2453-62. doi: 10.1016/j.ejmech.2011.03.030. Epub 2011 Mar 23. Eur J Med Chem. 2011. PMID: 21481497 Free PMC article.

10

N-Hydroxyindole-based inhibitors of lactate dehydrogenase against cancer cell proliferation.

Granchi C, Roy S, De Simone A, Salvetti I, Tuccinardi T, Martinelli A, Macchia M, Lanza M, Betti L, Giannaccini G, Lucacchini A, Giovannetti E, Sciarrillo R, Peters GJ, Minutolo F. Granchi C, et al. Eur J Med Chem. 2011 Nov;46(11):5398-407. doi: 10.1016/j.ejmech.2011.08.046. Epub 2011 Sep 8. Eur J Med Chem. 2011. PMID: 21944286

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