Kiss R - Search Results

1

3D-QSAR, design, synthesis and characterization of trisubstituted harmine derivatives with in vitro antiproliferative properties.

Meinguet C, Bruyère C, Frédérick R, Mathieu V, Vancraeynest C, Pochet L, Laloy J, Mortier J, Wolber G, Kiss R, Masereel B, Wouters J. Meinguet C, et al. Among authors: kiss r. Eur J Med Chem. 2015 Apr 13;94:45-55. doi: 10.1016/j.ejmech.2015.02.044. Epub 2015 Feb 24. Eur J Med Chem. 2015. PMID: 25747498 Free article.

2

N-(2-{3-[3,5-bis(trifluoromethyl)phenyl]ureido}ethyl)-glycyrrhetinamide (6b): a novel anticancer glycyrrhetinic acid derivative that targets the proteasome and displays anti-kinase activity.

Lallemand B, Chaix F, Bury M, Bruyère C, Ghostin J, Becker JP, Delporte C, Gelbcke M, Mathieu V, Dubois J, Prévost M, Jabin I, Kiss R. Lallemand B, et al. Among authors: kiss r. J Med Chem. 2011 Oct 13;54(19):6501-13. doi: 10.1021/jm200285z. Epub 2011 Sep 2. J Med Chem. 2011. PMID: 21888390

3

Novel trisubstituted harmine derivatives with original in vitro anticancer activity.

Frédérick R, Bruyère C, Vancraeynest C, Reniers J, Meinguet C, Pochet L, Backlund A, Masereel B, Kiss R, Wouters J. Frédérick R, et al. Among authors: kiss r. J Med Chem. 2012 Jul 26;55(14):6489-501. doi: 10.1021/jm300542e. Epub 2012 Jul 18. J Med Chem. 2012. PMID: 22770529 Free article.

4

New 5-Aryl-1H-imidazoles display in vitro antitumor activity against apoptosis-resistant cancer models, including melanomas, through mitochondrial targeting.

Mathieu V, Van Den Berge E, Ceusters J, Konopka T, Cops A, Bruyère C, Pirker C, Berger W, Trieu-Van T, Serteyn D, Kiss R, Robiette R. Mathieu V, et al. Among authors: kiss r. J Med Chem. 2013 Sep 12;56(17):6626-37. doi: 10.1021/jm400287v. Epub 2013 Aug 20. J Med Chem. 2013. PMID: 23845202

5

Growth inhibitory activity for cancer cell lines of lapachol and its natural and semi-synthetic derivatives.

Fiorito S, Epifano F, Bruyère C, Mathieu V, Kiss R, Genovese S. Fiorito S, et al. Among authors: kiss r. Bioorg Med Chem Lett. 2014 Jan 15;24(2):454-7. doi: 10.1016/j.bmcl.2013.12.049. Epub 2013 Dec 18. Bioorg Med Chem Lett. 2014. PMID: 24374273

6

New imidazo[1,2-b]pyrazoles as anticancer agents: synthesis, biological evaluation and structure activity relationship analysis.

Grosse S, Mathieu V, Pillard C, Massip S, Marchivie M, Jarry C, Bernard P, Kiss R, Guillaumet G. Grosse S, et al. Among authors: kiss r. Eur J Med Chem. 2014 Sep 12;84:718-30. doi: 10.1016/j.ejmech.2014.07.057. Epub 2014 Jul 18. Eur J Med Chem. 2014. PMID: 25064349

7

A harmine-derived beta-carboline displays anti-cancer effects in vitro by targeting protein synthesis.

Carvalho A, Chu J, Meinguet C, Kiss R, Vandenbussche G, Masereel B, Wouters J, Kornienko A, Pelletier J, Mathieu V. Carvalho A, et al. Among authors: kiss r. Eur J Pharmacol. 2017 Jun 15;805:25-35. doi: 10.1016/j.ejphar.2017.03.034. Epub 2017 Mar 18. Eur J Pharmacol. 2017. PMID: 28322844 Free PMC article.

8

Structure-activity relationship analysis of novel derivatives of narciclasine (an Amaryllidaceae isocarbostyril derivative) as potential anticancer agents.

Ingrassia L, Lefranc F, Dewelle J, Pottier L, Mathieu V, Spiegl-Kreinecker S, Sauvage S, El Yazidi M, Dehoux M, Berger W, Van Quaquebeke E, Kiss R. Ingrassia L, et al. Among authors: kiss r. J Med Chem. 2009 Feb 26;52(4):1100-14. doi: 10.1021/jm8013585. J Med Chem. 2009. PMID: 19199649

9

Lycorine, the main phenanthridine Amaryllidaceae alkaloid, exhibits significant antitumor activity in cancer cells that display resistance to proapoptotic stimuli: an investigation of structure-activity relationship and mechanistic insight.

Lamoral-Theys D, Andolfi A, Van Goietsenoven G, Cimmino A, Le Calvé B, Wauthoz N, Mégalizzi V, Gras T, Bruyère C, Dubois J, Mathieu V, Kornienko A, Kiss R, Evidente A. Lamoral-Theys D, et al. Among authors: kiss r. J Med Chem. 2009 Oct 22;52(20):6244-56. doi: 10.1021/jm901031h. J Med Chem. 2009. PMID: 19788245 Free PMC article.

10

Investigations of fungal secondary metabolites with potential anticancer activity.

Balde ES, Andolfi A, Bruyère C, Cimmino A, Lamoral-Theys D, Vurro M, Damme MV, Altomare C, Mathieu V, Kiss R, Evidente A. Balde ES, et al. Among authors: kiss r. J Nat Prod. 2010 May 28;73(5):969-71. doi: 10.1021/np900731p. J Nat Prod. 2010. PMID: 20415482

Save citations to file

Email citations

Send citations to clipboard

Add to Collections

Add to My Bibliography

Create a file for external citation management software

Your saved search

Your RSS Feed

My Custom Filters

Publication date

Text availability

Article attribute

Article type

Article Language

Species

Sex

Age

Other

1,011 results

Search Page

Filters