Mortier J - Search Results

1

3D-QSAR, design, synthesis and characterization of trisubstituted harmine derivatives with in vitro antiproliferative properties.

Meinguet C, Bruyère C, Frédérick R, Mathieu V, Vancraeynest C, Pochet L, Laloy J, Mortier J, Wolber G, Kiss R, Masereel B, Wouters J. Meinguet C, et al. Among authors: mortier j. Eur J Med Chem. 2015 Apr 13;94:45-55. doi: 10.1016/j.ejmech.2015.02.044. Epub 2015 Feb 24. Eur J Med Chem. 2015. PMID: 25747498 Free article.

2

Computational tools for in silico fragment-based drug design.

Mortier J, Rakers C, Frederick R, Wolber G. Mortier J, et al. Curr Top Med Chem. 2012;12(17):1935-43. doi: 10.2174/156802612804547371. Curr Top Med Chem. 2012. PMID: 23116473 Review.

3

Design, synthesis and structure-activity relationship of novel quinoxaline derivatives as cancer chemopreventive agent by inhibition of tyrosine kinase receptor.

Galal SA, Abdelsamie AS, Soliman SM, Mortier J, Wolber G, Ali MM, Tokuda H, Suzuki N, Lida A, Ramadan RA, El Diwani HI. Galal SA, et al. Among authors: mortier j. Eur J Med Chem. 2013 Nov;69:115-24. doi: 10.1016/j.ejmech.2013.07.049. Epub 2013 Aug 13. Eur J Med Chem. 2013. PMID: 24013411

4

Design, synthesis and molecular docking study of novel quinoxalin-2(1H)-ones as anti-tumor active agents with inhibition of tyrosine kinase receptor and studying their cyclooxygenase-2 activity.

Galal SA, Khairat SH, Ragab FA, Abdelsamie AS, Ali MM, Soliman SM, Mortier J, Wolber G, El Diwani HI. Galal SA, et al. Among authors: mortier j. Eur J Med Chem. 2014 Oct 30;86:122-32. doi: 10.1016/j.ejmech.2014.08.048. Epub 2014 Aug 15. Eur J Med Chem. 2014. PMID: 25147154

5

NF-kappaB inducing kinase (NIK) inhibitors: identification of new scaffolds using virtual screening.

Mortier J, Masereel B, Remouchamps C, Ganeff C, Piette J, Frederick R. Mortier J, et al. Bioorg Med Chem Lett. 2010 Aug 1;20(15):4515-20. doi: 10.1016/j.bmcl.2010.06.027. Epub 2010 Jun 8. Bioorg Med Chem Lett. 2010. PMID: 20580552

6

Synthesis, biological activity and structure-activity relationships of new benzoic acid-based protein tyrosine phosphatase inhibitors endowed with insulinomimetic effects in mouse C2C12 skeletal muscle cells.

Ottanà R, Maccari R, Mortier J, Caselli A, Amuso S, Camici G, Rotondo A, Wolber G, Paoli P. Ottanà R, et al. Among authors: mortier j. Eur J Med Chem. 2014 Jan;71:112-27. doi: 10.1016/j.ejmech.2013.11.001. Epub 2013 Nov 11. Eur J Med Chem. 2014. PMID: 24287560

7

From carbohydrates to drug-like fragments: Rational development of novel α-amylase inhibitors.

Al-Asri J, Fazekas E, Lehoczki G, Perdih A, Görick C, Melzig MF, Gyémánt G, Wolber G, Mortier J. Al-Asri J, et al. Among authors: mortier j. Bioorg Med Chem. 2015 Oct 15;23(20):6725-32. doi: 10.1016/j.bmc.2015.09.007. Epub 2015 Sep 8. Bioorg Med Chem. 2015. PMID: 26395057

8

Pyrazolo[4,3-c]isoquinolines as potential inhibitors of NF-kappaB activation.

Mortier J, Frederick R, Ganeff C, Remouchamps C, Talaga P, Pochet L, Wouters J, Piette J, Dejardin E, Masereel B. Mortier J, et al. Biochem Pharmacol. 2010 May 15;79(10):1462-72. doi: 10.1016/j.bcp.2010.01.007. Epub 2010 Jan 21. Biochem Pharmacol. 2010. PMID: 20096267

9

Inhibitory potency of flavonoid derivatives on influenza virus neuraminidase.

Rakers C, Schwerdtfeger SM, Mortier J, Duwe S, Wolff T, Wolber G, Melzig MF. Rakers C, et al. Among authors: mortier j. Bioorg Med Chem Lett. 2014 Sep 1;24(17):4312-7. doi: 10.1016/j.bmcl.2014.07.010. Epub 2014 Jul 18. Bioorg Med Chem Lett. 2014. PMID: 25096296

10

The impact of molecular dynamics on drug design: applications for the characterization of ligand-macromolecule complexes.

Mortier J, Rakers C, Bermudez M, Murgueitio MS, Riniker S, Wolber G. Mortier J, et al. Drug Discov Today. 2015 Jun;20(6):686-702. doi: 10.1016/j.drudis.2015.01.003. Epub 2015 Jan 20. Drug Discov Today. 2015. PMID: 25615716 Review.

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