Frehland B - Search Results

1

Stereoselective synthesis and pharmacological evaluation of [4.3.3]propellan-8-amines as analogs of adamantanamines.

Torres-Gómez H, Lehmkuhl K, Frehland B, Daniliuc C, Schepmann D, Ehrhardt C, Wünsch B. Torres-Gómez H, et al. Among authors: frehland b. Bioorg Med Chem. 2015 Aug 1;23(15):4277-4285. doi: 10.1016/j.bmc.2015.06.030. Epub 2015 Jun 18. Bioorg Med Chem. 2015. PMID: 26145819

2

Design, Synthesis, and Biological Evaluation of 3-Benzazepin-1-ols as NR2B-Selective NMDA Receptor Antagonists.

Tewes B, Frehland B, Schepmann D, Schmidtke KU, Winckler T, Wünsch B. Tewes B, et al. Among authors: frehland b. ChemMedChem. 2010 May 3;5(5):687-95. doi: 10.1002/cmdc.201000005. ChemMedChem. 2010. PMID: 20340125

3

Development of a selective competitive receptor binding assay for the determination of the affinity to NR2B containing NMDA receptors.

Schepmann D, Frehland B, Lehmkuhl K, Tewes B, Wünsch B. Schepmann D, et al. Among authors: frehland b. J Pharm Biomed Anal. 2010 Nov 2;53(3):603-8. doi: 10.1016/j.jpba.2010.04.014. Epub 2010 Apr 18. J Pharm Biomed Anal. 2010. PMID: 20462722

4

Conformationally constrained NR2B selective NMDA receptor antagonists derived from ifenprodil: Synthesis and biological evaluation of tetrahydro-3-benzazepine-1,7-diols.

Tewes B, Frehland B, Schepmann D, Schmidtke KU, Winckler T, Wünsch B. Tewes B, et al. Among authors: frehland b. Bioorg Med Chem. 2010 Nov 15;18(22):8005-15. doi: 10.1016/j.bmc.2010.09.026. Epub 2010 Sep 24. Bioorg Med Chem. 2010. PMID: 20965739

5

Characterization of ligand binding to the σ(1) receptor in a human tumor cell line (RPMI 8226) and establishment of a competitive receptor binding assay.

Brune S, Schepmann D, Lehmkuhl K, Frehland B, Wünsch B. Brune S, et al. Among authors: frehland b. Assay Drug Dev Technol. 2012 Aug;10(4):365-74. doi: 10.1089/adt.2011.0376. Epub 2011 Dec 22. Assay Drug Dev Technol. 2012. PMID: 22192304

6

Hydroxyalkylation with cyclic sulfates: synthesis of carbazole derived CB(2) ligands with increased polarity.

Lueg C, Galla F, Frehland B, Schepmann D, Daniliuc CG, Deuther-Conrad W, Brust P, Wünsch B. Lueg C, et al. Among authors: frehland b. Arch Pharm (Weinheim). 2014 Jan;347(1):21-31. doi: 10.1002/ardp.201300255. Epub 2013 Nov 18. Arch Pharm (Weinheim). 2014. PMID: 24243315

7

Synthesis, σ receptor affinity, and pharmacological evaluation of 5-phenylsulfanyl- and 5-benzyl-substituted tetrahydro-2-benzazepines.

Hasebein P, Frehland B, Schepmann D, Wünsch B. Hasebein P, et al. Among authors: frehland b. ChemMedChem. 2014 Aug;9(8):1697-703. doi: 10.1002/cmdc.201402110. Epub 2014 Jun 4. ChemMedChem. 2014. PMID: 24895069

8

Synthesis and pharmacological evaluation of like- and unlike-configured tetrahydro-2-benzazepines with the α-substituted benzyl moiety in the 5-position.

Hasebein P, Frehland B, Lehmkuhl K, Fröhlich R, Schepmann D, Wünsch B. Hasebein P, et al. Among authors: frehland b. Org Biomol Chem. 2014 Aug 7;12(29):5407-26. doi: 10.1039/c4ob00510d. Org Biomol Chem. 2014. PMID: 24934693

9

Synthesis, binding affinity and structure-activity relationships of novel, selective and dual targeting CCR2 and CCR5 receptor antagonists.

Junker A, Kokornaczyk AK, Zweemer AJ, Frehland B, Schepmann D, Yamaguchi J, Itami K, Faust A, Hermann S, Wagner S, Schäfers M, Koch M, Weiss C, Heitman LH, Kopka K, Wünsch B. Junker A, et al. Among authors: frehland b. Org Biomol Chem. 2015 Feb 28;13(8):2407-22. doi: 10.1039/c4ob02397h. Org Biomol Chem. 2015. PMID: 25566983

10

Enantiomerically Pure 2-Methyltetrahydro-3-benzazepin-1-ols Selectively Blocking GluN2B Subunit Containing N-Methyl-D-aspartate Receptors.

Tewes B, Frehland B, Schepmann D, Robaa D, Uengwetwanit T, Gaube F, Winckler T, Sippl W, Wünsch B. Tewes B, et al. Among authors: frehland b. J Med Chem. 2015 Aug 13;58(15):6293-305. doi: 10.1021/acs.jmedchem.5b00897. Epub 2015 Jul 30. J Med Chem. 2015. PMID: 26186074

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