Chavan A - Search Results

1

Discovery of Azaindole Ureas as a Novel Class of Bacterial Gyrase B Inhibitors.

Zhang J, Yang Q, Cross JB, Romero JA, Poutsiaka KM, Epie F, Bevan D, Wang B, Zhang Y, Chavan A, Zhang X, Moy T, Daniel A, Nguyen K, Chamberlain B, Carter N, Shotwell J, Silverman J, Metcalf CA 3rd, Ryan D, Lippa B, Dolle RE. Zhang J, et al. Among authors: chavan a. J Med Chem. 2015 Nov 12;58(21):8503-12. doi: 10.1021/acs.jmedchem.5b00961. Epub 2015 Oct 22. J Med Chem. 2015. PMID: 26460684

2

Structure-based discovery of LpxC inhibitors.

Zhang J, Chan A, Lippa B, Cross JB, Liu C, Yin N, Romero JA, Lawrence J, Heney R, Herradura P, Goss J, Clark C, Abel C, Zhang Y, Poutsiaka KM, Epie F, Conrad M, Mahamoon A, Nguyen K, Chavan A, Clark E, Li TC, Cheng RK, Wood M, Andersen OA, Brooks M, Kwong J, Barker J, Parr IB, Gu Y, Ryan MD, Coleman S, Metcalf CA 3rd. Zhang J, et al. Among authors: chavan a. Bioorg Med Chem Lett. 2017 Apr 15;27(8):1670-1680. doi: 10.1016/j.bmcl.2017.03.006. Epub 2017 Mar 6. Bioorg Med Chem Lett. 2017. PMID: 28302397

3

Novel A,B,E-ring-modified camptothecins displaying high lipophilicity and markedly improved human blood stabilities.

Bom D, Curran DP, Chavan AJ, Kruszewski S, Zimmer SG, Fraley KA, Burke TG. Bom D, et al. Among authors: chavan aj. J Med Chem. 1999 Aug 12;42(16):3018-22. doi: 10.1021/jm9902279. J Med Chem. 1999. PMID: 10447944 No abstract available.

4

Photoaffinity labeling of human placental NAD(+)-linked 15-hydroxyprostaglandin dehydrogenase with [alpha-32P]2N3NAD+. Identification of a peptide in the adenine ring binding domain.

Chavan AJ, Ensor CM, Wu P, Haley BE, Tai HH. Chavan AJ, et al. J Biol Chem. 1993 Aug 5;268(22):16437-42. J Biol Chem. 1993. PMID: 8344929 Free article.

5

Forskolin photoaffinity probes for the evaluation of tubulin binding sites.

Chavan AJ, Richardson SK, Kim H, Haley BE, Watt DS. Chavan AJ, et al. Bioconjug Chem. 1993 Jul-Aug;4(4):268-74. doi: 10.1021/bc00022a004. Bioconjug Chem. 1993. PMID: 8218483 No abstract available.

6

A photoactive phosphonamide derivative of GTP for the identification of the GTP-binding domain in beta-tubulin.

Chavan AJ, Kim H, Haley BE, Watt DS. Chavan AJ, et al. Bioconjug Chem. 1990 Sep-Oct;1(5):337-44. doi: 10.1021/bc00005a007. Bioconjug Chem. 1990. PMID: 2098111

7

The novel silatecan 7-tert-butyldimethylsilyl-10-hydroxycamptothecin displays high lipophilicity, improved human blood stability, and potent anticancer activity.

Bom D, Curran DP, Kruszewski S, Zimmer SG, Thompson Strode J, Kohlhagen G, Du W, Chavan AJ, Fraley KA, Bingcang AL, Latus LJ, Pommier Y, Burke TG. Bom D, et al. Among authors: chavan aj. J Med Chem. 2000 Oct 19;43(21):3970-80. doi: 10.1021/jm000144o. J Med Chem. 2000. PMID: 11052802

8

Synthesis and application of bidentate photoaffinity cross-linking reagents. Nucleotide photoaffinity probes with two photoactive groups.

Rajagopalan K, Chavan AJ, Haley BE, Watt DS. Rajagopalan K, et al. Among authors: chavan aj. J Biol Chem. 1993 Jul 5;268(19):14230-8. J Biol Chem. 1993. PMID: 8314786 Free article.

9

Modification of adenylate cyclase by photoaffinity analogs of forskolin.

Ho LT, Nie ZM, Mende TJ, Richardson S, Chavan A, Kolaczkowska E, Watt DS, Haley BE, Ho RJ. Ho LT, et al. Among authors: chavan a. Second Messengers Phosphoproteins. 1988-1989;12(5-6):209-23. Second Messengers Phosphoproteins. 1988. PMID: 3272297

10

Inhibition of granulocyte-macrophage colony-stimulating factor (GM-CSF) activity by suramin and suramin analogues is correlated to interaction with the GM-CSF nucleotide-binding site.

Doukas M, Chavan A, Gass C, Nickel P, Boone T, Haley B. Doukas M, et al. Among authors: chavan a. Cancer Res. 1995 Nov 15;55(22):5161-3. Cancer Res. 1995. PMID: 7585565

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