Kassiou M - Search Results

1

Pharmacology of novel small-molecule tubulin inhibitors in glioblastoma cells with enhanced EGFR signalling.

Phoa AF, Browne S, Gurgis FM, Åkerfeldt MC, Döbber A, Renn C, Peifer C, Stringer BW, Day BW, Wong C, Chircop M, Johns TG, Kassiou M, Munoz L. Phoa AF, et al. Among authors: kassiou m. Biochem Pharmacol. 2015 Dec 15;98(4):587-601. doi: 10.1016/j.bcp.2015.10.014. Epub 2015 Oct 28. Biochem Pharmacol. 2015. PMID: 26519552

2

Optimisation of LRRK2 inhibitors and assessment of functional efficacy in cell-based models of neuroinflammation.

Munoz L, Kavanagh ME, Phoa AF, Heng B, Dzamko N, Chen EJ, Doddareddy MR, Guillemin GJ, Kassiou M. Munoz L, et al. Among authors: kassiou m. Eur J Med Chem. 2015 May 5;95:29-34. doi: 10.1016/j.ejmech.2015.03.003. Epub 2015 Mar 3. Eur J Med Chem. 2015. PMID: 25791676

3

DYRK1A in neurodegeneration and cancer: Molecular basis and clinical implications.

Abbassi R, Johns TG, Kassiou M, Munoz L. Abbassi R, et al. Among authors: kassiou m. Pharmacol Ther. 2015 Jul;151:87-98. doi: 10.1016/j.pharmthera.2015.03.004. Epub 2015 Mar 17. Pharmacol Ther. 2015. PMID: 25795597 Review.

4

TSPO as a target for glioblastoma therapeutics.

Werry EL, Barron ML, Kassiou M. Werry EL, et al. Among authors: kassiou m. Biochem Soc Trans. 2015 Aug;43(4):531-6. doi: 10.1042/BST20150015. Epub 2015 Aug 3. Biochem Soc Trans. 2015. PMID: 26551689 Review.

5

Derivatives of the pyrazolo[1,5-a]pyrimidine acetamide DPA-713 as translocator protein (TSPO) ligands and pro-apoptotic agents in human glioblastoma.

Werry EL, King VA, Barron ML, Banister SD, Sokias R, Kassiou M. Werry EL, et al. Among authors: kassiou m. Eur J Pharm Sci. 2017 Jan 1;96:186-192. doi: 10.1016/j.ejps.2016.09.026. Epub 2016 Sep 19. Eur J Pharm Sci. 2017. PMID: 27658888

6

Kinase targets in CNS drug discovery.

Gunosewoyo H, Yu L, Munoz L, Kassiou M. Gunosewoyo H, et al. Among authors: kassiou m. Future Med Chem. 2017 Mar;9(3):303-314. doi: 10.4155/fmc-2016-0214. Epub 2017 Feb 8. Future Med Chem. 2017. PMID: 28176536

7

Structural Optimization and Pharmacological Evaluation of Inhibitors Targeting Dual-Specificity Tyrosine Phosphorylation-Regulated Kinases (DYRK) and CDC-like kinases (CLK) in Glioblastoma.

Zhou Q, Phoa AF, Abbassi RH, Hoque M, Reekie TA, Font JS, Ryan RM, Stringer BW, Day BW, Johns TG, Munoz L, Kassiou M. Zhou Q, et al. Among authors: kassiou m. J Med Chem. 2017 Mar 9;60(5):2052-2070. doi: 10.1021/acs.jmedchem.6b01840. Epub 2017 Feb 28. J Med Chem. 2017. PMID: 28206758

8

Discovery and pharmacological evaluation of a novel series of adamantyl cyanoguanidines as P2X₇ receptor antagonists.

O'Brien-Brown J, Jackson A, Reekie TA, Barron ML, Werry EL, Schiavini P, McDonnell M, Munoz L, Wilkinson S, Noll B, Wang S, Kassiou M. O'Brien-Brown J, et al. Among authors: kassiou m. Eur J Med Chem. 2017 Apr 21;130:433-439. doi: 10.1016/j.ejmech.2017.02.060. Epub 2017 Mar 2. Eur J Med Chem. 2017. PMID: 28279849

9

Changes in cell morphology guide identification of tubulin as the off-target for protein kinase inhibitors.

Hoque M, Abbassi RH, Froio D, Man J, Johns TG, Stringer BW, Day BW, Pajic M, Kassiou M, Munoz L. Hoque M, et al. Among authors: kassiou m. Pharmacol Res. 2018 Aug;134:166-178. doi: 10.1016/j.phrs.2018.06.023. Epub 2018 Jun 23. Pharmacol Res. 2018. PMID: 29944980

10

Determination and reduction of translocator protein (TSPO) ligand rs6971 discrimination.

Sokias R, Werry EL, Chua SW, Reekie TA, Munoz L, Wong ECN, Ittner LM, Kassiou M. Sokias R, et al. Among authors: kassiou m. Medchemcomm. 2016 Nov 15;8(1):202-210. doi: 10.1039/c6md00523c. eCollection 2017 Jan 1. Medchemcomm. 2016. PMID: 30108706 Free PMC article.

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