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23 results

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Page 1
Identification of pyrazolopyridazinones as PDEδ inhibitors.
Papke B, Murarka S, Vogel HA, Martín-Gago P, Kovacevic M, Truxius DC, Fansa EK, Ismail S, Zimmermann G, Heinelt K, Schultz-Fademrecht C, Al Saabi A, Baumann M, Nussbaumer P, Wittinghofer A, Waldmann H, Bastiaens PI. Papke B, et al. Among authors: fansa ek. Nat Commun. 2016 Apr 20;7:11360. doi: 10.1038/ncomms11360. Nat Commun. 2016. PMID: 27094677 Free PMC article.
Structure-based development of PDEδ inhibitors.
Martín-Gago P, Fansa EK, Wittinghofer A, Waldmann H. Martín-Gago P, et al. Among authors: fansa ek. Biol Chem. 2017 May 1;398(5-6):535-545. doi: 10.1515/hsz-2016-0272. Biol Chem. 2017. PMID: 27935847 Free article. Review.
Development of Pyridazinone Chemotypes Targeting the PDEδ Prenyl Binding Site.
Murarka S, Martín-Gago P, Schultz-Fademrecht C, Al Saabi A, Baumann M, Fansa EK, Ismail S, Nussbaumer P, Wittinghofer A, Waldmann H. Murarka S, et al. Among authors: fansa ek. Chemistry. 2017 May 2;23(25):6083-6093. doi: 10.1002/chem.201603222. Epub 2016 Nov 3. Chemistry. 2017. PMID: 27809361
The N- and C-terminal ends of RPGR can bind to PDE6δ.
Fansa EK, O'Reilly NJ, Ismail S, Wittinghofer A. Fansa EK, et al. EMBO Rep. 2015 Dec;16(12):1583-5. doi: 10.15252/embr.201541404. Epub 2015 Nov 9. EMBO Rep. 2015. PMID: 26553937 Free PMC article.
Sorting of lipidated cargo by the Arl2/Arl3 system.
Fansa EK, Wittinghofer A. Fansa EK, et al. Small GTPases. 2016 Oct;7(4):222-230. doi: 10.1080/21541248.2016.1224454. Epub 2016 Nov 2. Small GTPases. 2016. PMID: 27806215 Free PMC article. Review.
A PDE6δ-KRas Inhibitor Chemotype with up to Seven H-Bonds and Picomolar Affinity that Prevents Efficient Inhibitor Release by Arl2.
Martín-Gago P, Fansa EK, Klein CH, Murarka S, Janning P, Schürmann M, Metz M, Ismail S, Schultz-Fademrecht C, Baumann M, Bastiaens PI, Wittinghofer A, Waldmann H. Martín-Gago P, et al. Among authors: fansa ek. Angew Chem Int Ed Engl. 2017 Feb 20;56(9):2423-2428. doi: 10.1002/anie.201610957. Epub 2017 Jan 20. Angew Chem Int Ed Engl. 2017. PMID: 28106325
Covalent Protein Labeling at Glutamic Acids.
Martín-Gago P, Fansa EK, Winzker M, Murarka S, Janning P, Schultz-Fademrecht C, Baumann M, Wittinghofer A, Waldmann H. Martín-Gago P, et al. Among authors: fansa ek. Cell Chem Biol. 2017 May 18;24(5):589-597.e5. doi: 10.1016/j.chembiol.2017.03.015. Epub 2017 Apr 20. Cell Chem Biol. 2017. PMID: 28434875 Free article.
Small-Molecule Inhibition of the UNC119-Cargo Interaction.
Mejuch T, Garivet G, Hofer W, Kaiser N, Fansa EK, Ehrt C, Koch O, Baumann M, Ziegler S, Wittinghofer A, Waldmann H. Mejuch T, et al. Among authors: fansa ek. Angew Chem Int Ed Engl. 2017 May 22;56(22):6181-6186. doi: 10.1002/anie.201701905. Epub 2017 May 4. Angew Chem Int Ed Engl. 2017. PMID: 28471079
23 results