Georg G - Search Results

1

Inducing Protein Degradation as a Therapeutic Strategy.

Crews CM, Georg G, Wang S. Crews CM, et al. Among authors: georg g. J Med Chem. 2016 Jun 9;59(11):5129-30. doi: 10.1021/acs.jmedchem.6b00735. Epub 2016 May 20. J Med Chem. 2016. PMID: 27199030 No abstract available.

2

Synthesis of biologically active taxol analogues with modified phenylisoserine side chains.

Georg GI, Cheruvallath ZS, Himes RH, Mejillano MR, Burke CT. Georg GI, et al. J Med Chem. 1992 Oct 30;35(22):4230-7. doi: 10.1021/jm00100a031. J Med Chem. 1992. PMID: 1359143

3

Novel cytotoxic 3'-(tert-butyl) 3'-dephenyl analogs of paclitaxel and docetaxel.

Ali SM, Hoemann MZ, Aubé J, Mitscher LA, Georg GI, McCall R, Jayasinghe LR. Ali SM, et al. Among authors: georg gi. J Med Chem. 1995 Sep 15;38(19):3821-8. doi: 10.1021/jm00019a012. J Med Chem. 1995. PMID: 7562913

4

The effect of the aromatic rings of taxol on biological activity and solution conformation: synthesis and evaluation of saturated taxol and taxotere analogues.

Boge TC, Himes RH, Vander Velde DG, Georg GI. Boge TC, et al. Among authors: georg gi. J Med Chem. 1994 Sep 30;37(20):3337-43. doi: 10.1021/jm00046a018. J Med Chem. 1994. PMID: 7932561

5

4-Deacetyltaxol and 10-acetyl-4-deacetyltaxotere: synthesis and biological evaluation.

Datta A, Jayasinghe LR, Georg GI. Datta A, et al. Among authors: georg gi. J Med Chem. 1994 Nov 25;37(24):4258-60. doi: 10.1021/jm00050a023. J Med Chem. 1994. PMID: 7990125

6

Preparation of phenolic paclitaxel metabolites.

Park H, Hepperle M, Boge TC, Himes RH, Georg GI. Park H, et al. Among authors: georg gi. J Med Chem. 1996 Jul 5;39(14):2705-9. doi: 10.1021/jm960142x. J Med Chem. 1996. PMID: 8709100

7

Butitaxel analogues: synthesis and structure-activity relationships.

Ali SM, Hoemann MZ, Aubé J, Georg GI, Mitscher LA, Jayasinghe LR. Ali SM, et al. Among authors: georg gi. J Med Chem. 1997 Jan 17;40(2):236-41. doi: 10.1021/jm960505t. J Med Chem. 1997. PMID: 9003522

8

Total synthesis and evaluation of C25-benzyloxyepothilone C for tubulin assembly and cytotoxicity against MCF-7 breast cancer cells.

Hutt OE, Reddy BS, Nair SK, Reiff EA, Henri JT, Greiner JF, Chiu TL, Vandervelde DG, Amin EA, Himes RH, Georg GI. Hutt OE, et al. Among authors: georg gi. Bioorg Med Chem Lett. 2008 Sep 1;18(17):4904-6. doi: 10.1016/j.bmcl.2008.07.024. Epub 2008 Jul 11. Bioorg Med Chem Lett. 2008. PMID: 18684624 Free PMC article.

9

Paclitaxel succinate analogs: Anionic and amide introduction as a strategy to impart blood-brain barrier permeability.

Turunen BJ, Ge H, Oyetunji J, Desino KE, Vasandani V, Güthe S, Himes RH, Audus KL, Seelig A, Georg GI. Turunen BJ, et al. Bioorg Med Chem Lett. 2008 Nov 15;18(22):5971-4. doi: 10.1016/j.bmcl.2008.09.103. Epub 2008 Oct 2. Bioorg Med Chem Lett. 2008. PMID: 18926701 Free PMC article.

10

Synthesis, tubulin assembly, and antiproliferative activity against MCF7 and NCI/ADR-RES cancer cells of 10-O-acetyl-5'-hydroxybutitaxel.

Ge H, Wang J, Kayser MM, Himes RH, Georg GI. Ge H, et al. Bioorg Med Chem Lett. 2008 Dec 1;18(23):6165-7. doi: 10.1016/j.bmcl.2008.10.010. Epub 2008 Oct 7. Bioorg Med Chem Lett. 2008. PMID: 18977659 Free PMC article.

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