Hartmann RW - Search Results

1

Discovery and Structure-Based Optimization of 2-Ureidothiophene-3-carboxylic Acids as Dual Bacterial RNA Polymerase and Viral Reverse Transcriptase Inhibitors.

Elgaher WA, Sharma KK, Haupenthal J, Saladini F, Pires M, Real E, Mély Y, Hartmann RW. Elgaher WA, et al. Among authors: hartmann rw. J Med Chem. 2016 Aug 11;59(15):7212-22. doi: 10.1021/acs.jmedchem.6b00730. Epub 2016 Jul 7. J Med Chem. 2016. PMID: 27339173

2

Tetrahydronaphthalenes: influence of heterocyclic substituents on inhibition of steroid enzymes P450 arom and P450 17.

Wächter GA, Hartmann RW, Sergejew T, Grün GL, Ledergerber D. Wächter GA, et al. Among authors: hartmann rw. J Med Chem. 1996 Feb 16;39(4):834-41. doi: 10.1021/jm950377t. J Med Chem. 1996. PMID: 8632407

3

Imidazole substituted biphenyls: a new class of highly potent and in vivo active inhibitors of P450 17 as potential therapeutics for treatment of prostate cancer.

Wachall BG, Hector M, Zhuang Y, Hartmann RW. Wachall BG, et al. Among authors: hartmann rw. Bioorg Med Chem. 1999 Sep;7(9):1913-24. doi: 10.1016/s0968-0896(99)00160-1. Bioorg Med Chem. 1999. PMID: 10530940

4

Synthesis of N-substituted piperidine-4-(benzylidene-4-carboxylic acids) and evaluation as inhibitors of steroid-5alpha-reductase type 1 and 2.

Picard F, Baston E, Reichert W, Hartmann RW. Picard F, et al. Among authors: hartmann rw. Bioorg Med Chem. 2000 Jun;8(6):1479-87. doi: 10.1016/s0968-0896(00)00070-5. Bioorg Med Chem. 2000. PMID: 10896124

5

Synthesis and evaluation of novel steroidal oxime inhibitors of P450 17 (17 alpha-hydroxylase/C17-20-lyase) and 5 alpha-reductase types 1 and 2.

Hartmann RW, Hector M, Haidar S, Ehmer PB, Reichert W, Jose J. Hartmann RW, et al. J Med Chem. 2000 Nov 2;43(22):4266-77. doi: 10.1021/jm001008m. J Med Chem. 2000. PMID: 11063622

6

Synthesis and evaluation of 17-aliphatic heterocycle-substituted steroidal inhibitors of 17alpha-hydroxylase/C17-20-lyase (P450 17).

Hartmann RW, Hector M, Wachall BG, Palusczak A, Palzer M, Huch V, Veith M. Hartmann RW, et al. J Med Chem. 2000 Nov 16;43(23):4437-45. doi: 10.1021/jm991070n. J Med Chem. 2000. PMID: 11087568

7

A new class of nonsteroidal aromatase inhibitors: design and synthesis of chromone and xanthone derivatives and inhibition of the P450 enzymes aromatase and 17 alpha-hydroxylase/C17,20-lyase.

Recanatini M, Bisi A, Cavalli A, Belluti F, Gobbi S, Rampa A, Valenti P, Palzer M, Palusczak A, Hartmann RW. Recanatini M, et al. Among authors: hartmann rw. J Med Chem. 2001 Mar 1;44(5):672-80. doi: 10.1021/jm000955s. J Med Chem. 2001. PMID: 11262078

8

5-Phenyl substituted 1-methyl-2-pyridones and 4'-substituted biphenyl-4-carboxylic acids. synthesis and evaluation as inhibitors of steroid-5alpha-reductase type 1 and 2.

Picard F, Schulz T, Hartmann RW. Picard F, et al. Among authors: hartmann rw. Bioorg Med Chem. 2002 Feb;10(2):437-48. doi: 10.1016/s0968-0896(01)00293-0. Bioorg Med Chem. 2002. PMID: 11741792

9

Synthesis and evaluation of 2'-substituted 4-(4'-carboxy- or 4'-carboxymethylbenzylidene)-N-acylpiperidines: highly potent and in vivo active steroid 5alpha-reductase type 2 inhibitors.

Picard F, Barassin S, Mokhtarian A, Hartmann RW. Picard F, et al. Among authors: hartmann rw. J Med Chem. 2002 Aug 1;45(16):3406-17. doi: 10.1021/jm0208471. J Med Chem. 2002. PMID: 12139451

10

N-substituted 4-(4-carboxyphenoxy)benzamides. Synthesis and evaluation as inhibitors of steroid-5alpha-reductase type 1 and 2.

Picard F, Hartmann RW. Picard F, et al. Among authors: hartmann rw. J Enzyme Inhib Med Chem. 2002 Jun;17(3):187-96. doi: 10.1080/1475636021000003156. J Enzyme Inhib Med Chem. 2002. PMID: 12443045 Free article.

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