Rovira X - Search Results

1

OptoGluNAM4.1, a Photoswitchable Allosteric Antagonist for Real-Time Control of mGlu4 Receptor Activity.

Rovira X, Trapero A, Pittolo S, Zussy C, Faucherre A, Jopling C, Giraldo J, Pin JP, Gorostiza P, Goudet C, Llebaria A. Rovira X, et al. Cell Chem Biol. 2016 Aug 18;23(8):929-34. doi: 10.1016/j.chembiol.2016.06.013. Epub 2016 Jul 28. Cell Chem Biol. 2016. PMID: 27478159 Free article.

2

The catalytic power of enzymes: conformational selection or transition state stabilization?

Giraldo J, Roche D, Rovira X, Serra J. Giraldo J, et al. Among authors: rovira x. FEBS Lett. 2006 Apr 17;580(9):2170-7. doi: 10.1016/j.febslet.2006.03.060. Epub 2006 Mar 30. FEBS Lett. 2006. PMID: 16616138 Free article.

3

Assessing receptor affinity for inverse agonists: Schild and Cheng-Prusoff methods revisited.

Giraldo J, Serra J, Roche D, Rovira X. Giraldo J, et al. Among authors: rovira x. Curr Drug Targets. 2007 Jan;8(1):197-202. doi: 10.2174/138945007779315687. Curr Drug Targets. 2007. PMID: 17266542 Review.

4

Modeling the binding and function of metabotropic glutamate receptors.

Rovira X, Roche D, Serra J, Kniazeff J, Pin JP, Giraldo J. Rovira X, et al. J Pharmacol Exp Ther. 2008 May;325(2):443-56. doi: 10.1124/jpet.107.133967. Epub 2008 Feb 20. J Pharmacol Exp Ther. 2008. PMID: 18287211 Free article.

5

Modelling the interdependence between the stoichiometry of receptor oligomerization and ligand binding for a coexisting dimer/tetramer receptor system.

Rovira X, Vivó M, Serra J, Roche D, Strange PG, Giraldo J. Rovira X, et al. Br J Pharmacol. 2009 Jan;156(1):28-35. doi: 10.1111/j.1476-5381.2008.00031.x. Br J Pharmacol. 2009. PMID: 19133989 Free PMC article. Review.

6

The asymmetric/symmetric activation of GPCR dimers as a possible mechanistic rationale for multiple signalling pathways.

Rovira X, Pin JP, Giraldo J. Rovira X, et al. Trends Pharmacol Sci. 2010 Jan;31(1):15-21. doi: 10.1016/j.tips.2009.10.008. Epub 2009 Dec 4. Trends Pharmacol Sci. 2010. PMID: 19963287 Review.

7

An allosteric modulator to control endogenous G protein-coupled receptors with light.

Pittolo S, Gómez-Santacana X, Eckelt K, Rovira X, Dalton J, Goudet C, Pin JP, Llobet A, Giraldo J, Llebaria A, Gorostiza P. Pittolo S, et al. Among authors: rovira x. Nat Chem Biol. 2014 Oct;10(10):813-5. doi: 10.1038/nchembio.1612. Epub 2014 Aug 31. Nat Chem Biol. 2014. PMID: 25173999

8

Exploring the active conformation of cyclohexane carboxylate positive allosteric modulators of the type 4 metabotropic glutamate receptor.

Rovira X, Harrak Y, Trapero A, González-Bulnes P, Malhaire F, Pin JP, Goudet C, Giraldo J, Llebaria A. Rovira X, et al. ChemMedChem. 2014 Dec;9(12):2685-98. doi: 10.1002/cmdc.201402190. Epub 2014 Sep 5. ChemMedChem. 2014. PMID: 25196639

9

Overlapping binding sites drive allosteric agonism and positive cooperativity in type 4 metabotropic glutamate receptors.

Rovira X, Malhaire F, Scholler P, Rodrigo J, Gonzalez-Bulnes P, Llebaria A, Pin JP, Giraldo J, Goudet C. Rovira X, et al. FASEB J. 2015 Jan;29(1):116-30. doi: 10.1096/fj.14-257287. Epub 2014 Oct 23. FASEB J. 2015. PMID: 25342125

10

Major ligand-induced rearrangement of the heptahelical domain interface in a GPCR dimer.

Xue L, Rovira X, Scholler P, Zhao H, Liu J, Pin JP, Rondard P. Xue L, et al. Among authors: rovira x. Nat Chem Biol. 2015 Feb;11(2):134-40. doi: 10.1038/nchembio.1711. Epub 2014 Dec 15. Nat Chem Biol. 2015. PMID: 25503927

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