(R)-PFI-2 is a potent and selective inhibitor of SETD7 methyltransferase activity in cells.
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Barsyte-Lovejoy D, et al. Among authors: gingras ac.
Proc Natl Acad Sci U S A. 2014 Sep 2;111(35):12853-8. doi: 10.1073/pnas.1407358111. Epub 2014 Aug 18.
Proc Natl Acad Sci U S A. 2014.
PMID: 25136132
Free PMC article.