Cadavid MI - Search Results

1

Enantiospecific Recognition at the A_2B Adenosine Receptor by Alkyl 2-Cyanoimino-4-substituted-6-methyl-1,2,3,4-tetrahydropyrimidine-5-carboxylates.

Carbajales C, Azuaje J, Oliveira A, Loza MI, Brea J, Cadavid MI, Masaguer CF, García-Mera X, Gutiérrez-de-Terán H, Sotelo E. Carbajales C, et al. Among authors: cadavid mi. J Med Chem. 2017 Apr 27;60(8):3372-3382. doi: 10.1021/acs.jmedchem.7b00138. Epub 2017 Apr 11. J Med Chem. 2017. PMID: 28368607

2

Effect of Nitrogen Atom Substitution in A₃ Adenosine Receptor Binding: N-(4,6-Diarylpyridin-2-yl)acetamides as Potent and Selective Antagonists.

Azuaje J, Jespers W, Yaziji V, Mallo A, Majellaro M, Caamaño O, Loza MI, Cadavid MI, Brea J, Åqvist J, Sotelo E, Gutiérrez-de-Terán H. Azuaje J, et al. Among authors: cadavid mi. J Med Chem. 2017 Sep 14;60(17):7502-7511. doi: 10.1021/acs.jmedchem.7b00860. Epub 2017 Aug 21. J Med Chem. 2017. PMID: 28792759

3

Synthesis, adenosine receptor binding and 3D-QSAR of 4-substituted 2-(2'-furyl)-1,2,4-triazolo[1,5-a]quinoxalines.

Martínez A, Gutiérrez-de-Terán H, Brea J, Raviña E, Loza MI, Cadavid MI, Sanz F, Vidal B, Segarra V, Sotelo E. Martínez A, et al. Among authors: cadavid mi. Bioorg Med Chem. 2008 Feb 15;16(4):2103-13. doi: 10.1016/j.bmc.2007.10.103. Epub 2008 Jan 24. Bioorg Med Chem. 2008. PMID: 18249548

4

Pyrimidine derivatives as potent and selective A3 adenosine receptor antagonists.

Yaziji V, Rodríguez D, Gutiérrez-de-Terán H, Coelho A, Caamaño O, García-Mera X, Brea J, Loza MI, Cadavid MI, Sotelo E. Yaziji V, et al. Among authors: cadavid mi. J Med Chem. 2011 Jan 27;54(2):457-71. doi: 10.1021/jm100843z. Epub 2010 Dec 27. J Med Chem. 2011. PMID: 21186795

5

Selective and potent adenosine A3 receptor antagonists by methoxyaryl substitution on the N-(2,6-diarylpyrimidin-4-yl)acetamide scaffold.

Yaziji V, Rodríguez D, Coelho A, García-Mera X, El Maatougui A, Brea J, Loza MI, Cadavid MI, Gutiérrez-de-Terán H, Sotelo E. Yaziji V, et al. Among authors: cadavid mi. Eur J Med Chem. 2013 Jan;59:235-42. doi: 10.1016/j.ejmech.2012.11.010. Epub 2012 Nov 24. Eur J Med Chem. 2013. PMID: 23231967

6

Discovery of 3,4-Dihydropyrimidin-2(1H)-ones As a Novel Class of Potent and Selective A2B Adenosine Receptor Antagonists.

Crespo A, El Maatougui A, Biagini P, Azuaje J, Coelho A, Brea J, Loza MI, Cadavid MI, García-Mera X, Gutiérrez-de-Terán H, Sotelo E. Crespo A, et al. Among authors: cadavid mi. ACS Med Chem Lett. 2013 Oct 3;4(11):1031-6. doi: 10.1021/ml400185v. eCollection 2013 Nov 14. ACS Med Chem Lett. 2013. PMID: 24900602 Free PMC article.

7

Design, synthesis, and structure-activity relationships of 1-,3-,8-, and 9-substituted-9-deazaxanthines at the human A2B adenosine receptor.

Carotti A, Cadavid MI, Centeno NB, Esteve C, Loza MI, Martinez A, Nieto R, Raviña E, Sanz F, Segarra V, Sotelo E, Stefanachi A, Vidal B. Carotti A, et al. Among authors: cadavid mi. J Med Chem. 2006 Jan 12;49(1):282-99. doi: 10.1021/jm0506221. J Med Chem. 2006. PMID: 16392813

8

1-, 3- and 8-substituted-9-deazaxanthines as potent and selective antagonists at the human A2B adenosine receptor.

Stefanachi A, Brea JM, Cadavid MI, Centeno NB, Esteve C, Loza MI, Martinez A, Nieto R, Raviña E, Sanz F, Segarra V, Sotelo E, Vidal B, Carotti A. Stefanachi A, et al. Among authors: cadavid mi. Bioorg Med Chem. 2008 Mar 15;16(6):2852-69. doi: 10.1016/j.bmc.2008.01.002. Epub 2008 Jan 10. Bioorg Med Chem. 2008. PMID: 18226909

9

Synthesis of novel 1-alkyl-8-substituted-3-(3-methoxypropyl) xanthines as putative A(2B) receptor antagonists.

Nieto MI, Balo MC, Brea J, Caamaño O, Cadavid MI, Fernández F, Mera XG, López C, Rodríguez-Borges JE. Nieto MI, et al. Among authors: cadavid mi. Bioorg Med Chem. 2009 May 1;17(9):3426-32. doi: 10.1016/j.bmc.2009.03.029. Epub 2009 Mar 21. Bioorg Med Chem. 2009. PMID: 19346133

10

Synthesis and allosteric modulation of the dopamine receptor by peptide analogs of L-prolyl-L-leucyl-glycinamide (PLG) modified in the L-proline or L-proline and L-leucine scaffolds.

Ferreira da Costa J, Caamaño O, Fernández F, García-Mera X, Sampaio-Dias IE, Brea JM, Cadavid MI. Ferreira da Costa J, et al. Among authors: cadavid mi. Eur J Med Chem. 2013 Nov;69:146-58. doi: 10.1016/j.ejmech.2013.08.001. Epub 2013 Aug 22. Eur J Med Chem. 2013. PMID: 24013414

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