Knapp S - Search Results

1

Discovery of a Selective Allosteric Inhibitor Targeting Macrodomain 2 of Polyadenosine-Diphosphate-Ribose Polymerase 14.

Schuller M, Riedel K, Gibbs-Seymour I, Uth K, Sieg C, Gehring AP, Ahel I, Bracher F, Kessler BM, Elkins JM, Knapp S. Schuller M, et al. Among authors: knapp s. ACS Chem Biol. 2017 Nov 17;12(11):2866-2874. doi: 10.1021/acschembio.7b00445. Epub 2017 Oct 19. ACS Chem Biol. 2017. PMID: 28991428 Free PMC article.

2

Doing more than just the structure-structural genomics in kinase drug discovery.

Marsden BD, Knapp S. Marsden BD, et al. Among authors: knapp s. Curr Opin Chem Biol. 2008 Feb;12(1):40-5. doi: 10.1016/j.cbpa.2008.01.042. Epub 2008 Feb 29. Curr Opin Chem Biol. 2008. PMID: 18267130 Review.

3

Structure of dystrophia myotonica protein kinase.

Elkins JM, Amos A, Niesen FH, Pike AC, Fedorov O, Knapp S. Elkins JM, et al. Among authors: knapp s. Protein Sci. 2009 Apr;18(4):782-91. doi: 10.1002/pro.82. Protein Sci. 2009. PMID: 19309729 Free PMC article.

4

Specific CLK inhibitors from a novel chemotype for regulation of alternative splicing.

Fedorov O, Huber K, Eisenreich A, Filippakopoulos P, King O, Bullock AN, Szklarczyk D, Jensen LJ, Fabbro D, Trappe J, Rauch U, Bracher F, Knapp S. Fedorov O, et al. Among authors: knapp s. Chem Biol. 2011 Jan 28;18(1):67-76. doi: 10.1016/j.chembiol.2010.11.009. Chem Biol. 2011. PMID: 21276940 Free PMC article.

5

Crystal structures of ABL-related gene (ABL2) in complex with imatinib, tozasertib (VX-680), and a type I inhibitor of the triazole carbothioamide class.

Salah E, Ugochukwu E, Barr AJ, von Delft F, Knapp S, Elkins JM. Salah E, et al. Among authors: knapp s. J Med Chem. 2011 Apr 14;54(7):2359-67. doi: 10.1021/jm101506n. Epub 2011 Mar 18. J Med Chem. 2011. PMID: 21417343 Free PMC article.

6

Analysis of conditions affecting auto-phosphorylation of human kinases during expression in bacteria.

Shrestha A, Hamilton G, O'Neill E, Knapp S, Elkins JM. Shrestha A, et al. Among authors: knapp s. Protein Expr Purif. 2012 Jan;81(1):136-143. doi: 10.1016/j.pep.2011.09.012. Epub 2011 Oct 1. Protein Expr Purif. 2012. PMID: 21985771 Free PMC article.

7

7,8-dichloro-1-oxo-β-carbolines as a versatile scaffold for the development of potent and selective kinase inhibitors with unusual binding modes.

Huber K, Brault L, Fedorov O, Gasser C, Filippakopoulos P, Bullock AN, Fabbro D, Trappe J, Schwaller J, Knapp S, Bracher F. Huber K, et al. Among authors: knapp s. J Med Chem. 2012 Jan 12;55(1):403-13. doi: 10.1021/jm201286z. Epub 2012 Jan 3. J Med Chem. 2012. PMID: 22136433 Free PMC article.

8

Benzodiazepines and benzotriazepines as protein interaction inhibitors targeting bromodomains of the BET family.

Filippakopoulos P, Picaud S, Fedorov O, Keller M, Wrobel M, Morgenstern O, Bracher F, Knapp S. Filippakopoulos P, et al. Among authors: knapp s. Bioorg Med Chem. 2012 Mar 15;20(6):1878-86. doi: 10.1016/j.bmc.2011.10.080. Epub 2011 Nov 4. Bioorg Med Chem. 2012. PMID: 22137933 Free PMC article.

9

The structure of the full-length tetrameric PKA regulatory RIIβ complex reveals the mechanism of allosteric PKA activation.

Elkins JM, Knapp S. Elkins JM, et al. Among authors: knapp s. Sci Signal. 2012 May 15;5(224):pe21. doi: 10.1126/scisignal.2003053. Sci Signal. 2012. PMID: 22589386

10

Fragment screening of cyclin G-associated kinase by weak affinity chromatography.

Meiby E, Knapp S, Elkins JM, Ohlson S. Meiby E, et al. Among authors: knapp s. Anal Bioanal Chem. 2012 Nov;404(8):2417-25. doi: 10.1007/s00216-012-6335-6. Epub 2012 Aug 24. Anal Bioanal Chem. 2012. PMID: 22918538 Free PMC article.

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