The small molecule CLP257 does not modify activity of the K+-Cl- co-transporter KCC2 but does potentiate GABAA receptor activity.
Cardarelli RA, Jones K, Pisella LI, Wobst HJ, McWilliams LJ, Sharpe PM, Burnham MP, Baker DJ, Chudotvorova I, Guyot J, Silayeva L, Morrow DH, Dekker N, Zicha S, Davies PA, Holenz J, Duggan ME, Dunlop J, Mather RJ, Wang Q, Medina I, Brandon NJ, Deeb TZ, Moss SJ.
Cardarelli RA, et al. Among authors: chudotvorova i.
Nat Med. 2017 Dec 7;23(12):1394-1396. doi: 10.1038/nm.4442.
Nat Med. 2017.
PMID: 29216042
Free PMC article.
No abstract available.