Sałat K - Search Results

1

The Magic of Crystal Structure-Based Inhibitor Optimization: Development of a Butyrylcholinesterase Inhibitor with Picomolar Affinity and in Vivo Activity.

Košak U, Brus B, Knez D, Žakelj S, Trontelj J, Pišlar A, Šink R, Jukič M, Živin M, Podkowa A, Nachon F, Brazzolotto X, Stojan J, Kos J, Coquelle N, Sałat K, Colletier JP, Gobec S. Košak U, et al. Among authors: salat k. J Med Chem. 2018 Jan 11;61(1):119-139. doi: 10.1021/acs.jmedchem.7b01086. Epub 2017 Dec 22. J Med Chem. 2018. PMID: 29227101

2

2-Substituted 4-hydroxybutanamides as potential inhibitors of γ-aminobutyric acid transporters mGAT1-mGAT4: synthesis and biological evaluation.

Kowalczyk P, Sałat K, Höfner GC, Guzior N, Filipek B, Wanner KT, Kulig K. Kowalczyk P, et al. Among authors: salat k. Bioorg Med Chem. 2013 Sep 1;21(17):5154-67. doi: 10.1016/j.bmc.2013.06.038. Epub 2013 Jun 26. Bioorg Med Chem. 2013. PMID: 23859778

3

Synthesis, biological evaluation and structure-activity relationship of new GABA uptake inhibitors, derivatives of 4-aminobutanamides.

Kowalczyk P, Sałat K, Höfner GC, Mucha M, Rapacz A, Podkowa A, Filipek B, Wanner KT, Kulig K. Kowalczyk P, et al. Among authors: salat k. Eur J Med Chem. 2014 Aug 18;83:256-73. doi: 10.1016/j.ejmech.2014.06.024. Epub 2014 Jun 12. Eur J Med Chem. 2014. PMID: 24973660

4

Synthesis of new N-benzylpiperidine derivatives as cholinesterase inhibitors with β-amyloid anti-aggregation properties and beneficial effects on memory in vivo.

Więckowska A, Więckowski K, Bajda M, Brus B, Sałat K, Czerwińska P, Gobec S, Filipek B, Malawska B. Więckowska A, et al. Among authors: salat k. Bioorg Med Chem. 2015 May 15;23(10):2445-57. doi: 10.1016/j.bmc.2015.03.051. Epub 2015 Mar 27. Bioorg Med Chem. 2015. PMID: 25868744

5

Anticonvulsant active inhibitor of GABA transporter subtype 1, tiagabine, with activity in mouse models of anxiety, pain and depression.

Sałat K, Podkowa A, Kowalczyk P, Kulig K, Dziubina A, Filipek B, Librowski T. Sałat K, et al. Pharmacol Rep. 2015 Jun;67(3):465-72. doi: 10.1016/j.pharep.2014.11.003. Epub 2014 Nov 21. Pharmacol Rep. 2015. PMID: 25933955

6

The effect of GABA transporter 1 (GAT1) inhibitor, tiagabine, on scopolamine-induced memory impairments in mice.

Sałat K, Podkowa A, Mogilski S, Zaręba P, Kulig K, Sałat R, Malikowska N, Filipek B. Sałat K, et al. Among authors: salat r. Pharmacol Rep. 2015 Dec;67(6):1155-62. doi: 10.1016/j.pharep.2015.04.018. Epub 2015 May 12. Pharmacol Rep. 2015. PMID: 26481535

7

The anxiolytic-like activity of a novel N-cycloalkyl-N-benzoylpiperazine derivative.

Strub DJ, Sałat K, Librowski T, Lochyński S, Gaweł M, Podkowa A. Strub DJ, et al. Among authors: salat k. Pharmacol Rep. 2016 Feb;68(1):62-5. doi: 10.1016/j.pharep.2015.06.139. Epub 2015 Jul 17. Pharmacol Rep. 2016. PMID: 26721353

8

Effect of pregabalin on contextual memory deficits and inflammatory state-related protein expression in streptozotocin-induced diabetic mice.

Sałat K, Gdula-Argasińska J, Malikowska N, Podkowa A, Lipkowska A, Librowski T. Sałat K, et al. Naunyn Schmiedebergs Arch Pharmacol. 2016 Jun;389(6):613-23. doi: 10.1007/s00210-016-1230-x. Epub 2016 Mar 17. Naunyn Schmiedebergs Arch Pharmacol. 2016. PMID: 26984821 Free PMC article.

9

Synthesis and anticonvulsant activities of novel 2-(cyclopentylmethylene)hydrazinyl-1,3-thiazoles in mouse models of seizures.

Łączkowski KZ, Sałat K, Misiura K, Podkowa A, Malikowska N. Łączkowski KZ, et al. Among authors: salat k. J Enzyme Inhib Med Chem. 2016 Dec;31(6):1576-82. doi: 10.3109/14756366.2016.1158172. Epub 2016 Apr 6. J Enzyme Inhib Med Chem. 2016. PMID: 27052195 Free article.

10

Antidepressant-like effects of scopolamine in mice are enhanced by the group II mGlu receptor antagonist LY341495.

Podkowa K, Podkowa A, Sałat K, Lenda T, Pilc A, Pałucha-Poniewiera A. Podkowa K, et al. Among authors: salat k. Neuropharmacology. 2016 Dec;111:169-179. doi: 10.1016/j.neuropharm.2016.08.031. Epub 2016 Aug 25. Neuropharmacology. 2016. PMID: 27569995

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