Talele TT - Search Results

1

Comprehensive Synthesis of Amino Acid-Derived Thiazole Peptidomimetic Analogues to Understand the Enigmatic Drug/Substrate-Binding Site of P-Glycoprotein.

Patel BA, Abel B, Barbuti AM, Velagapudi UK, Chen ZS, Ambudkar SV, Talele TT. Patel BA, et al. Among authors: talele tt. J Med Chem. 2018 Feb 8;61(3):834-864. doi: 10.1021/acs.jmedchem.7b01340. Epub 2018 Jan 23. J Med Chem. 2018. PMID: 29251928 Free PMC article.

2

3D-QSAR studies on malonyl coenzyme A decarboxylase inhibitors.

Patel MR, Talele TT. Patel MR, et al. Among authors: talele tt. Bioorg Med Chem. 2007 Jul 1;15(13):4470-81. doi: 10.1016/j.bmc.2007.04.025. Epub 2007 Apr 24. Bioorg Med Chem. 2007. PMID: 17482825

3

CoMFA and HQSAR studies on 6,7-dimethoxy-4-pyrrolidylquinazoline derivatives as phosphodiesterase10A inhibitors.

Kulkarni SS, Patel MR, Talele TT. Kulkarni SS, et al. Among authors: talele tt. Bioorg Med Chem. 2008 Apr 1;16(7):3675-86. doi: 10.1016/j.bmc.2008.02.013. Epub 2008 Feb 8. Bioorg Med Chem. 2008. PMID: 18299198

4

Design, synthesis and determination of antifungal activity of 5(6)-substituted benzotriazoles.

Patel PD, Patel MR, Kocsis B, Kocsis E, Graham SM, Warren AR, Nicholson SM, Billack B, Fronczek FR, Talele TT. Patel PD, et al. Among authors: talele tt. Eur J Med Chem. 2010 Jun;45(6):2214-22. doi: 10.1016/j.ejmech.2010.01.062. Epub 2010 Feb 6. Eur J Med Chem. 2010. PMID: 20181413

5

Structure-based virtual screening, synthesis and SAR of novel inhibitors of hepatitis C virus NS5B polymerase.

Talele TT, Arora P, Kulkarni SS, Patel MR, Singh S, Chudayeu M, Kaushik-Basu N. Talele TT, et al. Bioorg Med Chem. 2010 Jul 1;18(13):4630-8. doi: 10.1016/j.bmc.2010.05.030. Epub 2010 May 15. Bioorg Med Chem. 2010. PMID: 20627595 Free PMC article.

6

The synthesis of phenylalanine-derived C5-substituted rhodanines and their activity against selected methicillin-resistant Staphylococcus aureus (MRSA) strains.

Hardej D, Ashby CR Jr, Khadtare NS, Kulkarni SS, Singh S, Talele TT. Hardej D, et al. Among authors: talele tt. Eur J Med Chem. 2010 Dec;45(12):5827-32. doi: 10.1016/j.ejmech.2010.09.045. Epub 2010 Sep 25. Eur J Med Chem. 2010. PMID: 20947220

7

Sildenafil reverses ABCB1- and ABCG2-mediated chemotherapeutic drug resistance.

Shi Z, Tiwari AK, Shukla S, Robey RW, Singh S, Kim IW, Bates SE, Peng X, Abraham I, Ambudkar SV, Talele TT, Fu LW, Chen ZS. Shi Z, et al. Among authors: talele tt. Cancer Res. 2011 Apr 15;71(8):3029-41. doi: 10.1158/0008-5472.CAN-10-3820. Epub 2011 Mar 14. Cancer Res. 2011. PMID: 21402712 Free PMC article.

8

The phosphodiesterase-5 inhibitor vardenafil is a potent inhibitor of ABCB1/P-glycoprotein transporter.

Ding PR, Tiwari AK, Ohnuma S, Lee JW, An X, Dai CL, Lu QS, Singh S, Yang DH, Talele TT, Ambudkar SV, Chen ZS. Ding PR, et al. Among authors: talele tt. PLoS One. 2011 Apr 28;6(4):e19329. doi: 10.1371/journal.pone.0019329. PLoS One. 2011. PMID: 21552528 Free PMC article.

9

Blockade of Her2/neu binding to Hsp90 by emodin azide methyl anthraquinone derivative induces proteasomal degradation of Her2/neu.

Yan YY, Zheng LS, Zhang X, Chen LK, Singh S, Wang F, Zhang JY, Liang YJ, Dai CL, Gu LQ, Zeng MS, Talele TT, Chen ZS, Fu LW. Yan YY, et al. Among authors: talele tt. Mol Pharm. 2011 Oct 3;8(5):1687-97. doi: 10.1021/mp2000499. Epub 2011 Aug 17. Mol Pharm. 2011. PMID: 21812426

10

Synthesis and SAR optimization of diketo acid pharmacophore for HCV NS5B polymerase inhibition.

Bhatt A, Gurukumar KR, Basu A, Patel MR, Kaushik-Basu N, Talele TT. Bhatt A, et al. Among authors: talele tt. Eur J Med Chem. 2011 Oct;46(10):5138-45. doi: 10.1016/j.ejmech.2011.08.028. Epub 2011 Aug 26. Eur J Med Chem. 2011. PMID: 21893371 Free PMC article.

Save citations to file

Email citations

Send citations to clipboard

Add to Collections

Add to My Bibliography

Create a file for external citation management software

Your saved search

Your RSS Feed

My Custom Filters

Publication date

Text availability

Article attribute

Article type

Article Language

Species

Sex

Age

Other

98 results

Search Page

Filters