Christensen KE - Search Results

1

Synthesis of Novel Pyridine-Carboxylates as Small-Molecule Inhibitors of Human Aspartate/Asparagine-β-Hydroxylase.

Brewitz L, Tumber A, Thalhammer A, Salah E, Christensen KE, Schofield CJ. Brewitz L, et al. Among authors: christensen ke. ChemMedChem. 2020 Jul 3;15(13):1139-1149. doi: 10.1002/cmdc.202000147. Epub 2020 May 26. ChemMedChem. 2020. PMID: 32330361 Free PMC article.

2

2-Difluoromethoxy-Substituted Estratriene Sulfamates: Synthesis, Antiproliferative SAR, Antitubulin Activity, and Steroid Sulfatase Inhibition.

Dohle W, Asiki H, Gruchot W, Foster PA, Sahota HK, Bai R, Christensen KE, Hamel E, Potter BVL. Dohle W, et al. Among authors: christensen ke. ChemMedChem. 2022 Dec 5;17(23):e202200408. doi: 10.1002/cmdc.202200408. Epub 2022 Oct 13. ChemMedChem. 2022. PMID: 36109340 Free PMC article.

3

5-Substituted Pyridine-2,4-dicarboxylate Derivatives Have Potential for Selective Inhibition of Human Jumonji-C Domain-Containing Protein 5.

Brewitz L, Nakashima Y, Piasecka SK, Salah E, Fletcher SC, Tumber A, Corner TP, Kennedy TJ, Fiorini G, Thalhammer A, Christensen KE, Coleman ML, Schofield CJ. Brewitz L, et al. Among authors: christensen ke. J Med Chem. 2023 Aug 10;66(15):10849-10865. doi: 10.1021/acs.jmedchem.3c01114. Epub 2023 Aug 1. J Med Chem. 2023. PMID: 37527664 Free PMC article.

4

αβ,α'β'-Diepoxyketones are mechanism-based inhibitors of nucleophilic cysteine enzymes.

de Munnik M, Lithgow J, Brewitz L, Christensen KE, Bates RH, Rodriguez-Miquel B, Schofield CJ. de Munnik M, et al. Among authors: christensen ke. Chem Commun (Camb). 2023 Oct 26;59(86):12859-12862. doi: 10.1039/d3cc02932h. Chem Commun (Camb). 2023. PMID: 37815791 Free PMC article.

5

Controlling Intramolecular Interactions in the Design of Selective, High-Affinity Ligands for the CREBBP Bromodomain.

Brand M, Clayton J, Moroglu M, Schiedel M, Picaud S, Bluck JP, Skwarska A, Bolland H, Chan AKN, Laurin CMC, Scorah AR, See L, Rooney TPC, Andrews KH, Fedorov O, Perell G, Kalra P, Vinh KB, Cortopassi WA, Heitel P, Christensen KE, Cooper RI, Paton RS, Pomerantz WCK, Biggin PC, Hammond EM, Filippakopoulos P, Conway SJ. Brand M, et al. Among authors: christensen ke. J Med Chem. 2021 Jul 22;64(14):10102-10123. doi: 10.1021/acs.jmedchem.1c00348. Epub 2021 Jul 13. J Med Chem. 2021. PMID: 34255515 Free PMC article.

6

Enhancement of anion recognition exhibited by a halogen-bonding rotaxane host system.

Kilah NL, Wise MD, Serpell CJ, Thompson AL, White NG, Christensen KE, Beer PD. Kilah NL, et al. Among authors: christensen ke. J Am Chem Soc. 2010 Sep 1;132(34):11893-5. doi: 10.1021/ja105263q. J Am Chem Soc. 2010. PMID: 20687599

7

Synthesis and bioactivity of fused- and spiro-β-lactone-lactam systems.

Josa-Culleré L, Towers C, Willenbrock F, Macaulay VM, Christensen KE, Moloney MG. Josa-Culleré L, et al. Among authors: christensen ke. Org Biomol Chem. 2017 Jun 27;15(25):5373-5379. doi: 10.1039/c7ob01148b. Org Biomol Chem. 2017. PMID: 28617490

8

Convergent Total Syntheses of (-)-Rubriflordilactone B and (-)-pseudo-Rubriflordilactone B.

Mohammad M, Chintalapudi V, Carney JM, Mansfield SJ, Sanderson P, Christensen KE, Anderson EA. Mohammad M, et al. Among authors: christensen ke. Angew Chem Int Ed Engl. 2019 Dec 9;58(50):18177-18181. doi: 10.1002/anie.201908917. Epub 2019 Oct 31. Angew Chem Int Ed Engl. 2019. PMID: 31595605 Free PMC article.

9

Synthesis of Polysubstituted Fused Pyrroles by Gold-Catalyzed Cycloisomerization/1,2-Sulfonyl Migration of Yndiamides.

Smith PJ, Jiang Y, Tong Z, Pickford HD, Christensen KE, Nugent J, Anderson EA. Smith PJ, et al. Among authors: christensen ke. Org Lett. 2021 Aug 20;23(16):6547-6552. doi: 10.1021/acs.orglett.1c02360. Epub 2021 Aug 9. Org Lett. 2021. PMID: 34369785

10

Copper-Catalyzed Synthesis and Applications of Yndiamides.

Mansfield SJ, Christensen KE, Thompson AL, Ma K, Jones MW, Mekareeya A, Anderson EA. Mansfield SJ, et al. Among authors: christensen ke. Angew Chem Int Ed Engl. 2017 Nov 13;56(46):14428-14432. doi: 10.1002/anie.201706915. Epub 2017 Oct 13. Angew Chem Int Ed Engl. 2017. PMID: 28875510

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