Jacomini AP - Search Results

1

Synthesis of novel 3,5,6-trisubstituted 2-pyridone derivatives and evaluation for their anti-inflammatory activity.

Gonçalves DS, de S Melo SM, Jacomini AP, J V da Silva M, Pianoski KE, Ames FQ, Aguiar RP, Oliveira AF, Volpato H, Bidóia DL, Nakamura CV, Bersani-Amado CA, Back DF, Moura S, Paula FR, Rosa FA. Gonçalves DS, et al. Among authors: jacomini ap. Bioorg Med Chem. 2020 Jun 15;28(12):115549. doi: 10.1016/j.bmc.2020.115549. Epub 2020 May 12. Bioorg Med Chem. 2020. PMID: 32503692

2

Synthesis and evaluation against Leishmania amazonensis of novel pyrazolo[3,4-d]pyridazinone-N-acylhydrazone-(bi)thiophene hybrids.

Jacomini AP, Silva MJV, Silva RGM, Gonçalves DS, Volpato H, Basso EA, Paula FR, Nakamura CV, Sarragiotto MH, Rosa FA. Jacomini AP, et al. Eur J Med Chem. 2016 Nov 29;124:340-349. doi: 10.1016/j.ejmech.2016.08.048. Epub 2016 Aug 23. Eur J Med Chem. 2016. PMID: 27597410

3

Unconventional Method for Synthesis of 3-Carboxyethyl-4-formyl(hydroxy)-5-aryl-N-arylpyrazoles.

da Silva MJV, Poletto J, Jacomini AP, Pianoski KE, Gonçalves DS, Ribeiro GM, de S Melo SM, Back DF, Moura S, Rosa FA. da Silva MJV, et al. Among authors: jacomini ap. J Org Chem. 2017 Dec 1;82(23):12590-12602. doi: 10.1021/acs.joc.7b02361. Epub 2017 Nov 15. J Org Chem. 2017. PMID: 29094945

4

In vitro anti-Leishmania activity of T6 synthetic compound encapsulated in yeast-derived β-(1,3)-d-glucan particles.

Volpato H, Scariot DB, Soares EFP, Jacomini AP, Rosa FA, Sarragiotto MH, Ueda-Nakamura T, Rubira AF, Pereira GM, Manadas R, Leitão AJ, Borges O, Nakamura CV, Sousa MDC. Volpato H, et al. Among authors: jacomini ap. Int J Biol Macromol. 2018 Nov;119:1264-1275. doi: 10.1016/j.ijbiomac.2018.08.019. Epub 2018 Aug 7. Int J Biol Macromol. 2018. PMID: 30096400

5

One-Pot Highly Regioselective Synthesis of α-Ketoamide N-Arylpyrazoles from Secondary β-Enamino Diketones.

Poletto J, Ribeiro GM, da Silva MJV, Jacomini AP, Basso EA, Back DF, Moura S, Rosa FA. Poletto J, et al. Among authors: jacomini ap. Org Lett. 2019 Aug 16;21(16):6325-6328. doi: 10.1021/acs.orglett.9b02206. Epub 2019 Jul 29. Org Lett. 2019. PMID: 31353911

6

Oral treatment with T6-loaded yeast cell wall particles reduces the parasitemia in murine visceral leishmaniasis model.

Scariot DB, Volpato H, Fernandes NS, Lazarin-Bidóia D, Borges O, Sousa MDC, Rosa FA, Jacomini AP, Silva SO, Ueda-Nakamura T, Rubira AF, Nakamura CV. Scariot DB, et al. Among authors: jacomini ap. Sci Rep. 2019 Dec 27;9(1):20080. doi: 10.1038/s41598-019-56647-w. Sci Rep. 2019. PMID: 31882925 Free PMC article.

7

1,2-Addition to trifluoromethylated β-enamino diketones: regioselective synthesis of trifluoromethyl-containing azomethine pyrazoles and isoxazoles.

Pianoski KE, Poletto J, Vieira da Silva MJ, Ascencio Camargo JN, Jacomini AP, Gonçalves DS, Back DF, Moura S, Rosa FA. Pianoski KE, et al. Among authors: jacomini ap. Org Biomol Chem. 2020 Apr 1;18(13):2524-2537. doi: 10.1039/d0ob00319k. Org Biomol Chem. 2020. PMID: 32196053

8

Antiparasitic activities of novel pyrimidine N-acylhydrazone hybrids.

Poletto J, da Silva MJV, Jacomini AP, Bidóia DL, Volpato H, Nakamura CV, Rosa FA. Poletto J, et al. Among authors: jacomini ap. Drug Dev Res. 2021 Apr;82(2):230-240. doi: 10.1002/ddr.21745. Epub 2020 Sep 30. Drug Dev Res. 2021. PMID: 32996619

9

Efficient synthesis and antitumor evaluation of 4-aminomethyl-N-arylpyrazoles: Discovery of potent and selective agents for ovarian cancer.

da Silva MJV, Jacomini AP, Figueiredo MC, Back DF, Foglio MA, Ruiz ALTG, Paula FR, Rosa FA. da Silva MJV, et al. Among authors: jacomini ap. Bioorg Med Chem. 2021 Jan 1;29:115835. doi: 10.1016/j.bmc.2020.115835. Epub 2020 Nov 4. Bioorg Med Chem. 2021. PMID: 33214037 Free article.

10

Discovery of 1,3,4,5-tetrasubstituted pyrazoles as anti-trypanosomatid agents: Identification of alterations in flagellar structure of L. amazonensis.

da Silva MJV, Jacomini AP, Gonçalves DS, Pianoski KE, Poletto J, Lazarin-Bidóia D, Volpato H, Nakamura CV, Rosa FA. da Silva MJV, et al. Among authors: jacomini ap. Bioorg Chem. 2021 Sep;114:105082. doi: 10.1016/j.bioorg.2021.105082. Epub 2021 Jun 11. Bioorg Chem. 2021. PMID: 34147880

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