Brea J - Search Results

1

Correction to Bicyclic α-Iminophosphonates as High Affinity Imidazoline I₂ Receptor Ligands for Alzheimer's Disease.

Abás S, Rodríguez-Arévalo S, Bagán A, Griñán-Ferré C, Vasilopoulou F, Brocos-Mosquera I, Muguruza C, Pérez B, Molins E, Luque FJ, Pérez-Lozano P, de Jonghe S, Daelemans D, Naesens L, Brea J, Loza MI, Hernández-Hernández E, García-Sevilla JA, García-Fuster MJ, Radan M, Djikic T, Nikolic K, Pallàs M, Callado LF, Escolano C. Abás S, et al. Among authors: brea j. J Med Chem. 2020 Sep 24;63(18):10529. doi: 10.1021/acs.jmedchem.0c01324. Epub 2020 Sep 14. J Med Chem. 2020. PMID: 32924503 No abstract available.

2

Butyrophenone analogues in the carbazole series as potential atypical antipsychotics: synthesis and determination of affinities at D(2), 5-HT(2A), 5-HT(2B) and 5-HT(2C) receptors.

Masaguer CF, Raviña E, Fontenla JA, Brea J, Tristán H, Loza MI. Masaguer CF, et al. Among authors: brea j. Eur J Med Chem. 2000 Jan;35(1):83-95. doi: 10.1016/s0223-5234(00)00109-4. Eur J Med Chem. 2000. PMID: 10733606

3

New serotonin 5-HT(2A), 5-HT(2B), and 5-HT(2C) receptor antagonists: synthesis, pharmacology, 3D-QSAR, and molecular modeling of (aminoalkyl)benzo and heterocycloalkanones.

Brea J, Rodrigo J, Carrieri A, Sanz F, Cadavid MI, Enguix MJ, Villazón M, Mengod G, Caro Y, Masaguer CF, Raviña E, Centeno NB, Carotti A, Loza MI. Brea J, et al. J Med Chem. 2002 Jan 3;45(1):54-71. doi: 10.1021/jm011014y. J Med Chem. 2002. PMID: 11754579

4

New arylpiperazine derivatives with high affinity for alpha1A, D2 and 5-HT2A receptors.

González-Gómez JC, Santana L, Uriarte E, Brea J, Villazón M, Loza MI, De Luca M, Rivas ME, Montenegro GY, Fontenla JA. González-Gómez JC, et al. Among authors: brea j. Bioorg Med Chem Lett. 2003 Jan 20;13(2):175-8. doi: 10.1016/s0960-894x(02)00933-2. Bioorg Med Chem Lett. 2003. PMID: 12482418

5

Conformationally constrained butyrophenones as new pharmacological tools to study 5-HT 2A and 5-HT 2C receptor behaviours.

Brea J, Masaguer CF, Villazón M, Cadavid MI, Raviña E, Fontaine F, Dezi C, Pastor M, Sanz F, Loza MI. Brea J, et al. Eur J Med Chem. 2003 Apr;38(4):433-40. doi: 10.1016/s0223-5234(03)00054-0. Eur J Med Chem. 2003. PMID: 12750032

6

Chemoenzymatic synthesis and binding affinity of novel (R)- and (S)-3-aminomethyl-1-tetralones, potential atypical antipsychotics.

Caro Y, Torrado M, Masaguer CF, Raviña E, Padín F, Brea J, Loza MI. Caro Y, et al. Among authors: brea j. Bioorg Med Chem Lett. 2004 Feb 9;14(3):585-9. doi: 10.1016/j.bmcl.2003.11.064. Bioorg Med Chem Lett. 2004. PMID: 14741248

7

Synthesis and biological activity of new potential agonists for the human adenosine A2A receptor.

Bosch MP, Campos F, Niubó I, Rosell G, Díaz JL, Brea J, Loza MI, Guerrero A. Bosch MP, et al. Among authors: brea j. J Med Chem. 2004 Jul 29;47(16):4041-53. doi: 10.1021/jm031143+. J Med Chem. 2004. PMID: 15267242

8

Synthesis and binding affinity of novel 3-aminoethyl-1-tetralones, potential atypical antipsychotics.

Alvarado M, Coelho A, Masaguer CF, Raviña E, Brea J, Padín JF, Loza MI. Alvarado M, et al. Among authors: brea j. Bioorg Med Chem Lett. 2005 Jun 15;15(12):3063-6. doi: 10.1016/j.bmcl.2005.04.022. Bioorg Med Chem Lett. 2005. PMID: 15878662

9

Multistructure 3D-QSAR studies on a series of conformationally constrained butyrophenones docked into a new homology model of the 5-HT2A receptor.

Dezi C, Brea J, Alvarado M, Raviña E, Masaguer CF, Loza MI, Sanz F, Pastor M. Dezi C, et al. Among authors: brea j. J Med Chem. 2007 Jul 12;50(14):3242-55. doi: 10.1021/jm070277a. Epub 2007 Jun 19. J Med Chem. 2007. PMID: 17579386

10

Synthesis and binding affinity of new pyrazole and isoxazole derivatives as potential atypical antipsychotics.

Barceló M, Raviña E, Masaguer CF, Domínguez E, Areias FM, Brea J, Loza MI. Barceló M, et al. Among authors: brea j. Bioorg Med Chem Lett. 2007 Sep 1;17(17):4873-7. doi: 10.1016/j.bmcl.2007.06.045. Epub 2007 Jun 14. Bioorg Med Chem Lett. 2007. PMID: 17588750

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