Discovery of first-in-class inhibitors of ASH1L histone methyltransferase with anti-leukemic activity.
Rogawski DS, Deng J, Li H, Miao H, Borkin D, Purohit T, Song J, Chase J, Li S, Ndoj J, Klossowski S, Kim E, Mao F, Zhou B, Ropa J, Krotoska MZ, Jin Z, Ernst P, Feng X, Huang G, Nishioka K, Kelly S, He M, Wen B, Sun D, Muntean A, Dou Y, Maillard I, Cierpicki T, Grembecka J.
Rogawski DS, et al. Among authors: ropa j.
Nat Commun. 2021 May 14;12(1):2792. doi: 10.1038/s41467-021-23152-6.
Nat Commun. 2021.
PMID: 33990599
Free PMC article.